SCHEMBL5162372

SCHEMBL5162372

Cc1ccc(CC2(N(C)C)CCC(NC(=O)CCNC(=O)O)CC2)cc1

nearest known ligand 0.45

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 3/20 0.43
HPGD P15428 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
OPRM1 P35372 4/20 0.41
OPRL1 P41146 4/20 0.41
ALDH1A1 P00352 1/20 0.41
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
NPC1 O15118 2/20 0.38
KDM4E B2RXH2 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4075032 0.90 HPGD (0.40) RAB9AHPGDSMN1; SMN2OPRM1OPRL1
SCHEMBL206456 0.87 POLB (0.45) RAB9AHPGDSMN1; SMN2ALDH1A1KMT2A
SCHEMBL4869393 0.87 EPHX1 (0.42) RAB9AHPGDSMN1; SMN2OPRM1OPRL1
SCHEMBL4084293 0.86 HDAC3 (0.42) RAB9AHPGDSMN1; SMN2OPRM1OPRL1
SCHEMBL208660 0.85 PLAAT3 (0.46) RAB9ASMN1; SMN2OPRM1OPRL1NPC1
SCHEMBL206704 0.84 SMYD3 (0.39) RAB9AHPGDSMN1; SMN2ALDH1A1MEN1
SCHEMBL2983415 0.84 MEN1 (0.45) RAB9AHPGDSMN1; SMN2OPRM1OPRL1
SCHEMBL4048631 0.84 KMT2A (0.51) RAB9AOPRM1OPRL1ALDH1A1MEN1
SCHEMBL4084189 0.83 HRH3 (0.40) RAB9AHPGDSMN1; SMN2OPRM1OPRL1
SCHEMBL4072191 0.82 HPGD (0.38) RAB9AHPGDSMN1; SMN2OPRM1OPRL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1751090-A1 ACID DERIVATIVES OF SUBSTITUTED CYCLOHEXYL-1,4-DIAMINES Grünenthal GmbH (DE) 2007-02-14 EP disclosed
WO-2005110973-A1 ACID DERIVATIVES OF SUBSTITUTED CYCLOHEXYL-1,4-DIAMINES Grünenthal GmbH (DE) 2005-11-24 WO disclosed