SCHEMBL4072191

SCHEMBL4072191

Cc1ccc(CC2(N(C)C)CCC(NC(=O)CCC(=O)NCCNC(=O)C(F)(F)F)CC2)cc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 1/20 0.38
RAB9A P51151 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
ALDH1A1 P00352 2/20 0.37
OPRM1 P35372 2/20 0.36
OPRL1 P41146 2/20 0.36
HDAC3 O15379 2/20 0.36
HDAC1 Q13547 2/20 0.36
HDAC2 Q92769 2/20 0.36
HDAC6 Q9UBN7 2/20 0.36
HDAC4 P56524 1/20 0.36
HDAC7 Q8WUI4 1/20 0.36
HDAC10 Q969S8 1/20 0.36
HDAC11 Q96DB2 1/20 0.36
HDAC8 Q9BY41 1/20 0.36
HDAC9 Q9UKV0 1/20 0.36
HDAC5 Q9UQL6 1/20 0.36
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL209170 0.90 HPGD (0.35) HPGDRAB9ASMN1; SMN2ALDH1A1OPRM1
SCHEMBL206456 0.87 POLB (0.45) HPGDRAB9ASMN1; SMN2ALDH1A1KMT2A
SCHEMBL4075032 0.86 HPGD (0.40) HPGDRAB9ASMN1; SMN2ALDH1A1OPRM1
SCHEMBL205912 0.84 HPGD (0.47) HPGDRAB9AALDH1A1MEN1KMT2A
SCHEMBL4084293 0.84 HDAC3 (0.42) HPGDRAB9ASMN1; SMN2ALDH1A1OPRM1
SCHEMBL208660 0.83 PLAAT3 (0.46) RAB9ASMN1; SMN2OPRM1OPRL1
SCHEMBL207807 0.83 KMT2A (0.37) RAB9AALDH1A1OPRM1OPRL1MEN1
SCHEMBL206704 0.82 SMYD3 (0.39) HPGDRAB9ASMN1; SMN2ALDH1A1MEN1
SCHEMBL208300 0.82 LMNA (0.50) RAB9AALDH1A1MEN1KMT2A
SCHEMBL5162372 0.82 RAB9A (0.43) HPGDRAB9ASMN1; SMN2ALDH1A1OPRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1745010-B1 SUBSTITUTED CYCLOHEXYL-1,4-DIAMINE DERIVATIVES GRUENENTHAL GMBH (DE) 2009-08-05 EP claimed