SCHEMBL5162561

SCHEMBL5162561

CN(C)C1(CCc2ccccc2)CCC(NC(=O)C(Oc2cccc(Cl)c2)C(Oc2ccccc2)C(=O)NC2CCC(Cc3cccc(F)c3)(N(C)C)CC2)CC1

nearest known ligand 0.40

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.40
MAPT P10636 1/20 0.40
SIGMAR1 Q99720 4/20 0.38
PPARG P37231 1/20 0.38
PPARA Q07869 1/20 0.38
FFAR2 O15552 1/20 0.37
GHSR Q92847 2/20 0.37
OPRM1 P35372 3/20 0.37
OPRD1 P41143 1/20 0.37
KMT2A Q03164 2/20 0.35
POLB P06746 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5162540 0.86 MCHR1 (0.46) SIGMAR1POLB
SCHEMBL2989322 0.82 MEN1 (0.48) MAPTSIGMAR1PPARGPPARAOPRM1
SCHEMBL2976658 0.81 MEN1 (0.45) ALDH1A1MAPTSIGMAR1PPARGPPARA
SCHEMBL2984800 0.81 ALDH1A1 (0.48) ALDH1A1MAPTSIGMAR1FFAR2GHSR
SCHEMBL2982908 0.79 MCHR1 (0.50) SIGMAR1POLB
SCHEMBL2976726 0.77 MCHR1 (0.54) SIGMAR1POLB
SCHEMBL2972799 0.77 TSHR (0.52) ALDH1A1MAPTGHSROPRM1
SCHEMBL2987754 0.75 POLB (0.50) ALDH1A1SIGMAR1OPRM1KMT2APOLB
SCHEMBL2972810 0.75 ATF4 (0.55) SIGMAR1KMT2APOLB
SCHEMBL5162405 0.74 PPARG (0.39) ALDH1A1SIGMAR1PPARGPPARAKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2007536322-A 2007-12-13 JP claimed
EP-1747191-A1 SUBSTITUTED CYCLOHEXYL-1,4-DIAMINE DERIVATIVES WITH A CHAIN EXTENSION Grünenthal GmbH (DE) 2007-01-31 EP claimed
WO-2005110975-A1 SUBSTITUTED CYCLOHEXYL-1,4-DIAMINE DERIVATIVES WITH A CHAIN EXTENSION Grünenthal GmbH (DE) 2005-11-24 WO claimed