SCHEMBL5165079

SCHEMBL5165079

CN(C)C1(Cc2ccccc2)CCC(NCc2ccccc2)CC1

nearest known ligand 0.65

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 5/20 0.65
OPRL1 P41146 5/20 0.65
GRIN2B Q13224 4/20 0.51
OPRK1 P41145 1/20 0.51
ACHE P22303 3/20 0.48
BACE1 P56817 3/20 0.48
BCHE P06276 2/20 0.48
MEN1 O00255 2/20 0.47
KMT2A Q03164 2/20 0.47
RAB9A P51151 1/20 0.47
CARM1 Q86X55 1/20 0.46
PRMT6 Q96LA8 1/20 0.46
TMEM97 Q5BJF2 1/20 0.45
FABP6 P51161 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL5164761 0.98 OPRM1 (0.66) OPRM1OPRL1GRIN2BOPRK1ACHE
SCHEMBL5165779 0.88 OPRM1 (0.51) OPRM1OPRL1GRIN2BOPRK1
SCHEMBL5166242 0.85 OPRM1 (0.51) OPRM1OPRL1GRIN2BOPRK1MEN1
SCHEMBL5167763 0.84 OPRM1 (0.54) OPRM1OPRL1OPRK1
SCHEMBL5166608 0.80 OPRM1 (0.44) OPRM1OPRL1GRIN2BOPRK1
SCHEMBL5164787 0.80 OPRL1 (0.69) OPRM1OPRL1MEN1KMT2A
Hydrochloric Acid SCHEMBL5163755 0.80 OPRM1 (0.46) OPRM1OPRL1GRIN2BOPRK1
Hydrochloric Acid SCHEMBL5164262 0.80 OPRL1 (0.68) OPRM1OPRL1MEN1KMT2A
SCHEMBL21744620 0.79 OPRM1 (0.65) OPRM1OPRL1GRIN2BACHEBACE1
SCHEMBL14028057 0.79 OPRM1 (0.58) OPRM1OPRL1OPRK1ACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1392641-B1 SUBSTITUTED CYCLOHEXANE-1,4-DIAMINE DERIVATIVES GRUENENTHAL GMBH (DE) 2007-04-11 EP claimed
US-7276518-B2 Substituted cyclohexane-1,4-diamine compounds GRUENENTHAL GMBH (DE) 2007-10-02 US disclosed
EP-1392641-B1 SUBSTITUTED CYCLOHEXANE-1,4-DIAMINE DERIVATIVES GRUENENTHAL GMBH (DE) 2007-04-11 EP disclosed
US-20040229872-A1 Substituted cyclohexane-1,4-diamine compounds with anti-diarrhea and peripheral analgesic activity GRUENENTHAL GMBH (DE) 2004-11-18 US disclosed
US-20040162287-A1 Substituted cyclohexane-1,4-diamine compounds GRUENENTHAL GMBH (DE) 2004-08-19 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040162287-A1 Substituted cyclohexane-1,4-diamine compounds DPYD, DDC, QDPR OPRM1 459/4885OPRL1 1102/4885GRIN2B 1592/4885
US-20040229872-A1 Substituted cyclohexane-1,4-diamine compounds with anti-diarrhea and peripheral analgesic activity ARG1, CD2, PDCD1 OPRM1 250/4885OPRL1 41/4885GRIN2B 3244/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.