SCHEMBL5166238

SCHEMBL5166238

COc1cccc(C2(O)CCCN(CCOc3ccccc3)C2)c1

nearest known ligand 0.51

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.51
KMT2A Q03164 2/20 0.51
OPRM1 P35372 1/20 0.51
OPRD1 P41143 1/20 0.51
OPRK1 P41145 1/20 0.51
OPRL1 P41146 1/20 0.51
MEN1 O00255 1/20 0.51
LMNA P02545 1/20 0.51
LTA4H P09960 3/20 0.50
DRD2 P14416 3/20 0.49
KDM4E B2RXH2 1/20 0.47
ESR1 P03372 1/20 0.46
ESR2 Q92731 1/20 0.46
DRD3 P35462 1/20 0.45
GRIN2B Q13224 2/20 0.44
BACE1 P56817 1/20 0.44
HRH3 Q9Y5N1 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL3098282 0.99 ALDH1A1 (0.50) ALDH1A1KMT2AOPRM1OPRD1OPRK1
SCHEMBL5166952 0.87 HRH3 (0.55) ALDH1A1OPRM1OPRD1OPRK1OPRL1
Hydrochloric Acid SCHEMBL3085793 0.86 HRH3 (0.54) ALDH1A1OPRM1OPRD1OPRK1OPRL1
SCHEMBL3081018 0.84 ALDH1A1 (0.60) ALDH1A1KMT2AOPRM1OPRD1OPRK1
Hydrochloric Acid SCHEMBL11194779 0.83 ALDH1A1 (0.59) ALDH1A1KMT2AOPRM1OPRD1OPRK1
SCHEMBL5168106 0.82 OPRM1 (0.60) ALDH1A1KMT2AOPRM1OPRD1OPRK1
Hydrochloric Acid SCHEMBL3092573 0.81 OPRM1 (0.58) ALDH1A1KMT2AOPRM1OPRD1OPRK1
SCHEMBL17848367 0.81 MEN1 (0.58) ALDH1A1KMT2AOPRL1MEN1LMNA
SCHEMBL5166771 0.80 ALDH1A1 (0.60) ALDH1A1KMT2AOPRM1OPRD1OPRK1
SCHEMBL5165555 0.79 ALDH1A1 (0.54) ALDH1A1KMT2AOPRM1OPRD1OPRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1771417-A1 SUBSTITUTED 3-PHENYLPIPERIDINE DERIVATIVES Grünenthal GmbH (DE) 2007-04-11 EP claimed
WO-2006010577-A1 SUBSTITUTED 3-PHENYLPIPERIDINE DERIVATIVES Grünenthal GmbH (DE) 2006-02-02 WO claimed
EP-1771417-A1 SUBSTITUTED 3-PHENYLPIPERIDINE DERIVATIVES Grünenthal GmbH (DE) 2007-04-11 EP disclosed
WO-2006010577-A1 SUBSTITUTED 3-PHENYLPIPERIDINE DERIVATIVES Grünenthal GmbH (DE) 2006-02-02 WO disclosed