SCHEMBL5166952

SCHEMBL5166952

COc1cccc(C2(O)CCCN(CCc3ccccc3)C2)c1

nearest known ligand 0.56

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 1/20 0.55
SIGMAR1 Q99720 3/20 0.53
OPRM1 P35372 2/20 0.51
OPRD1 P41143 1/20 0.51
OPRK1 P41145 1/20 0.51
OPRL1 P41146 1/20 0.51
HTR1A P08908 1/20 0.50
SLC6A4 P31645 1/20 0.50
ALDH1A1 P00352 1/20 0.50
KCNH2 Q12809 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL3085793 0.99 HRH3 (0.54) HRH3SIGMAR1OPRM1OPRD1OPRK1
SCHEMBL3081018 0.89 ALDH1A1 (0.60) SIGMAR1OPRM1OPRD1OPRK1OPRL1
Hydrochloric Acid SCHEMBL11194779 0.88 ALDH1A1 (0.59) SIGMAR1OPRM1OPRD1OPRK1OPRL1
SCHEMBL5166238 0.87 ALDH1A1 (0.51) HRH3OPRM1OPRD1OPRK1OPRL1
Hydrochloric Acid SCHEMBL3098282 0.86 ALDH1A1 (0.50) HRH3OPRM1OPRD1OPRK1OPRL1
SCHEMBL7256584 0.84 SIGMAR1 (0.57) SIGMAR1OPRL1
Bromide SCHEMBL7248470 0.83 SIGMAR1 (0.56) SIGMAR1OPRL1
SCHEMBL5166185 0.83 ALDH1A1 (0.53) SIGMAR1OPRM1OPRD1OPRK1OPRL1
SCHEMBL5168106 0.82 OPRM1 (0.60) OPRM1OPRD1OPRK1OPRL1ALDH1A1
SCHEMBL5166771 0.82 ALDH1A1 (0.60) SIGMAR1OPRM1OPRD1OPRK1OPRL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1771417-A1 SUBSTITUTED 3-PHENYLPIPERIDINE DERIVATIVES Grünenthal GmbH (DE) 2007-04-11 EP claimed
WO-2006010577-A1 SUBSTITUTED 3-PHENYLPIPERIDINE DERIVATIVES Grünenthal GmbH (DE) 2006-02-02 WO claimed
EP-1771417-A1 SUBSTITUTED 3-PHENYLPIPERIDINE DERIVATIVES Grünenthal GmbH (DE) 2007-04-11 EP disclosed
WO-2006010577-A1 SUBSTITUTED 3-PHENYLPIPERIDINE DERIVATIVES Grünenthal GmbH (DE) 2006-02-02 WO disclosed