SCHEMBL5166883

SCHEMBL5166883

COc1cccc(C2(O)CCCN(Cc3cccc(C)c3)C2)c1

nearest known ligand 0.55

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MCHR1 Q99705 1/20 0.55
ALDH1A1 P00352 7/20 0.54
SIGMAR1 Q99720 1/20 0.46
MAPT P10636 1/20 0.46
MAPK1 P28482 1/20 0.46
NPSR1 Q6W5P4 1/20 0.46
GAA P10253 1/20 0.46
KMT2A Q03164 4/20 0.45
KDM4E B2RXH2 4/20 0.45
OPRM1 P35372 1/20 0.45
OPRD1 P41143 1/20 0.45
OPRK1 P41145 1/20 0.45
OPRL1 P41146 1/20 0.45
MEN1 O00255 3/20 0.44
HTR1D P28221 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
LMNA P02545 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL3091514 0.99 MCHR1 (0.54) MCHR1ALDH1A1SIGMAR1MAPTMAPK1
SCHEMBL5166618 0.90 ALDH1A1 (0.58) MCHR1ALDH1A1SIGMAR1MAPTMAPK1
SCHEMBL3081018 0.90 ALDH1A1 (0.60) ALDH1A1SIGMAR1KMT2AKDM4EOPRM1
Hydrochloric Acid SCHEMBL3074059 0.89 ALDH1A1 (0.57) MCHR1ALDH1A1SIGMAR1MAPTMAPK1
Hydrochloric Acid SCHEMBL11194779 0.89 ALDH1A1 (0.59) ALDH1A1SIGMAR1KMT2AKDM4EOPRM1
SCHEMBL5168656 0.88 ALDH1A1 (0.53) MCHR1ALDH1A1SIGMAR1GAAKMT2A
SCHEMBL5166185 0.88 ALDH1A1 (0.53) ALDH1A1SIGMAR1GAAKMT2AKDM4E
SCHEMBL5166771 0.88 ALDH1A1 (0.60) ALDH1A1SIGMAR1KMT2AKDM4EOPRM1
Hydrochloric Acid SCHEMBL3087862 0.87 ALDH1A1 (0.53) ALDH1A1SIGMAR1GAAKMT2AKDM4E
Hydrochloric Acid SCHEMBL3088477 0.87 ALDH1A1 (0.53) MCHR1ALDH1A1SIGMAR1GAAKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1771417-A1 SUBSTITUTED 3-PHENYLPIPERIDINE DERIVATIVES Grünenthal GmbH (DE) 2007-04-11 EP claimed
WO-2006010577-A1 SUBSTITUTED 3-PHENYLPIPERIDINE DERIVATIVES Grünenthal GmbH (DE) 2006-02-02 WO claimed
EP-1771417-A1 SUBSTITUTED 3-PHENYLPIPERIDINE DERIVATIVES Grünenthal GmbH (DE) 2007-04-11 EP disclosed
WO-2006010577-A1 SUBSTITUTED 3-PHENYLPIPERIDINE DERIVATIVES Grünenthal GmbH (DE) 2006-02-02 WO disclosed