SCHEMBL5168656

SCHEMBL5168656

COc1cccc(C2(O)CCCN(Cc3cccc(Br)c3)C2)c1

nearest known ligand 0.53

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.53
SMN1; SMN2 Q16637 1/20 0.48
TDP1 Q9NUW8 1/20 0.48
SIGMAR1 Q99720 1/20 0.45
GAA P10253 1/20 0.45
ALOX15 P16050 1/20 0.45
TSHR P16473 1/20 0.45
KDM4E B2RXH2 3/20 0.44
OPRM1 P35372 1/20 0.44
OPRD1 P41143 1/20 0.44
OPRK1 P41145 1/20 0.44
OPRL1 P41146 1/20 0.44
KMT2A Q03164 1/20 0.44
HTR1D P28221 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.43
MCHR1 Q99705 1/20 0.43
LMNA P02545 1/20 0.43
HTT P42858 1/20 0.43
MAOB P27338 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL3088477 0.99 ALDH1A1 (0.53) ALDH1A1SMN1; SMN2TDP1SIGMAR1GAA
SCHEMBL5168339 0.90 ALDH1A1 (0.57) ALDH1A1SMN1; SMN2SIGMAR1GAAALOX15
Hydrochloric Acid SCHEMBL3074049 0.89 ALDH1A1 (0.56) ALDH1A1SMN1; SMN2SIGMAR1ALOX15TSHR
SCHEMBL3081018 0.89 ALDH1A1 (0.60) ALDH1A1SIGMAR1TSHRKDM4EOPRM1
SCHEMBL5166883 0.88 MCHR1 (0.55) ALDH1A1SIGMAR1GAAKDM4EOPRM1
Hydrochloric Acid SCHEMBL11194779 0.88 ALDH1A1 (0.59) ALDH1A1SIGMAR1TSHRKDM4EOPRM1
SCHEMBL5166185 0.87 ALDH1A1 (0.53) ALDH1A1SMN1; SMN2SIGMAR1GAAKDM4E
Hydrochloric Acid SCHEMBL3091514 0.87 MCHR1 (0.54) ALDH1A1SIGMAR1GAAKDM4EOPRM1
SCHEMBL5166771 0.87 ALDH1A1 (0.60) ALDH1A1SMN1; SMN2SIGMAR1TSHRKDM4E
Hydrochloric Acid SCHEMBL3087862 0.86 ALDH1A1 (0.53) ALDH1A1SMN1; SMN2SIGMAR1GAAKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1771417-A1 SUBSTITUTED 3-PHENYLPIPERIDINE DERIVATIVES Grünenthal GmbH (DE) 2007-04-11 EP claimed
WO-2006010577-A1 SUBSTITUTED 3-PHENYLPIPERIDINE DERIVATIVES Grünenthal GmbH (DE) 2006-02-02 WO claimed
EP-1771417-A1 SUBSTITUTED 3-PHENYLPIPERIDINE DERIVATIVES Grünenthal GmbH (DE) 2007-04-11 EP disclosed
WO-2006010577-A1 SUBSTITUTED 3-PHENYLPIPERIDINE DERIVATIVES Grünenthal GmbH (DE) 2006-02-02 WO disclosed