SCHEMBL5167688

SCHEMBL5167688

Cc1ccc(C[C@]2(Nc3cnc(/C=C/C(=O)O)cn3)CCCNC2)cc1

nearest known ligand 0.38

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 13/20 0.32
AKR1C4 P17516 8/20 0.32
AKR1C2 P52895 8/20 0.32
AKR1C1 Q04828 4/20 0.32
LMNA P02545 1/20 0.32
SLC6A4 P31645 1/20 0.31
ADRA1A P35348 1/20 0.31
PTGS2 P35354 1/20 0.31
HRH1 P35367 1/20 0.31
OPRK1 P41145 1/20 0.31
ALDH1A1 P00352 1/20 0.30
ADRB2 P07550 1/20 0.30
HTT P42858 1/20 0.30
HDAC3 O15379 1/20 0.30
HDAC1 Q13547 1/20 0.30
HDAC2 Q92769 1/20 0.30
HDAC6 Q9UBN7 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5170237 0.94 AKR1C3 (0.33) AKR1C3AKR1C4AKR1C2AKR1C1LMNA
SCHEMBL5197780 0.91 HDAC3 (0.38) LMNASLC6A4ALDH1A1ADRB2HTT
SCHEMBL5169616 0.91 MAPKAPK2 (0.31) SLC6A4ALDH1A1ADRB2HTTHDAC3
SCHEMBL5171832 0.91 RAB9A (0.31) LMNAHRH1ALDH1A1ADRB2HTT
SCHEMBL5191421 0.85 HDAC3 (0.39) LMNASLC6A4ALDH1A1ADRB2HTT
SCHEMBL5170345 0.85
SCHEMBL5172911 0.85 HDAC1 (0.37) LMNAHDAC3HDAC1HDAC2HDAC6
SCHEMBL5195227 0.85 RAB9A (0.32) AKR1C3AKR1C4AKR1C2LMNAHRH1
SCHEMBL5195209 0.85 SLC6A2 (0.32) AKR1C3AKR1C4AKR1C2SLC6A4HDAC3
SCHEMBL5197786 0.84 SLC6A2 (0.36) LMNASLC6A4ALDH1A1HDAC3HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1776357-A1 HYDROXYAMIDE COMPOUNDS HAVING ACTIVITY AS INHIBITORS OF HISTONE DEACETYLASE (HDAC) Astellas Pharma Inc. (JP) 2007-04-25 EP disclosed
WO-2006016680-A1 HYDROXYAMIDE COMPOUNDS HAVING ACTIVITY AS INHIBITORS OF HISTONE DEACETYLASE (HDAC) ASTELLAS PHARMA INC. (JP) 2006-02-16 WO disclosed