SCHEMBL5168846

SCHEMBL5168846

Nc1cccc(C[C@@]2(NC(=O)O)CCNC2)c1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRM2 Q14416 1/20 0.37
GRM3 Q14832 1/20 0.37
SLC6A2 P23975 6/20 0.36
SLC6A4 P31645 6/20 0.36
SLC6A3 Q01959 6/20 0.36
CYP2D6 P10635 6/20 0.36
MAOA P21397 2/20 0.36
MAOB P27338 2/20 0.36
NAMPT P43490 1/20 0.35
HSD11B1 P28845 1/20 0.34
CHRM3 P20309 1/20 0.34
SSTR4 P31391 1/20 0.33
ROCK2 O75116 2/20 0.33
ALDH1A1 P00352 1/20 0.33
ADRB2 P07550 1/20 0.33
HTT P42858 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP2C9 P11712 1/20 0.33
TSHR P16473 1/20 0.33
CYP2C19 P33261 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5913507 0.85 MAOA (0.42) GRM2GRM3CYP2D6MAOAMAOB
SCHEMBL5171838 0.82 CYP2D6 (0.47) SLC6A2SLC6A4SLC6A3CYP2D6ALDH1A1
SCHEMBL5170529 0.82 HDAC1 (0.39) SLC6A2SLC6A4SLC6A3CYP2D6CHRM3
SCHEMBL5169163 0.81 KMT2A (0.42) CYP2D6MAOAMAOBALDH1A1CYP2C9
SCHEMBL5171729 0.81 NPSR1 (0.44) MAOBCHRM3ALDH1A1CYP1A2TSHR
SCHEMBL5170560 0.79 NR3C1 (0.40) ROCK2ALDH1A1ROCK1
SCHEMBL5167704 0.78 SMN1; SMN2 (0.39) SLC6A2SLC6A4SLC6A3CYP2D6ALDH1A1
SCHEMBL22499953 0.71 KDM4E (0.32)
SCHEMBL7972011 0.70 SLC6A2 (0.37) SLC6A2SLC6A4SLC6A3CYP2D6ALDH1A1
SCHEMBL1178048 0.69 MAOA (0.46) GRM2GRM3MAOAMAOBNAMPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1776357-A1 HYDROXYAMIDE COMPOUNDS HAVING ACTIVITY AS INHIBITORS OF HISTONE DEACETYLASE (HDAC) Astellas Pharma Inc. (JP) 2007-04-25 EP disclosed
WO-2006016680-A1 HYDROXYAMIDE COMPOUNDS HAVING ACTIVITY AS INHIBITORS OF HISTONE DEACETYLASE (HDAC) ASTELLAS PHARMA INC. (JP) 2006-02-16 WO disclosed