SCHEMBL5167704

SCHEMBL5167704

Cc1ccc(C[C@@]2(NC(=O)O)CCNC2)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.39
ADRB2 P07550 2/20 0.36
GABRD O14764 1/20 0.36
GABRA1 P14867 1/20 0.36
GABRB1 P18505 1/20 0.36
GABRA5 P31644 1/20 0.36
GABRA3 P34903 1/20 0.36
GABRA2 P47869 1/20 0.36
GABRB2 P47870 1/20 0.36
GABRA4 P48169 1/20 0.36
SLC6A2 P23975 6/20 0.36
SLC6A4 P31645 6/20 0.36
SLC6A3 Q01959 6/20 0.36
CYP2D6 P10635 5/20 0.36
ALDH1A1 P00352 3/20 0.36
HTT P42858 1/20 0.36
NPC1 O15118 2/20 0.35
MEN1 O00255 1/20 0.35
TP53 P04637 1/20 0.35
HPGD P15428 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5168846 0.78 GRM2 (0.37) ADRB2SLC6A2SLC6A4SLC6A3CYP2D6
SCHEMBL5170529 0.77 HDAC1 (0.39) SMN1; SMN2SLC6A2SLC6A4SLC6A3CYP2D6
SCHEMBL5171838 0.77 CYP2D6 (0.47) SMN1; SMN2SLC6A2SLC6A4SLC6A3CYP2D6
SCHEMBL5171729 0.76 NPSR1 (0.44) GABRDGABRA1GABRB1GABRA5GABRA3
SCHEMBL28060870 0.75 OPRM1 (0.33) KMT2A
SCHEMBL5170560 0.75 NR3C1 (0.40) SMN1; SMN2ALDH1A1
SCHEMBL1035119 0.74 PPIA (0.42) ADRB2SLC6A2SLC6A4SLC6A3CYP2D6
SCHEMBL5170237 0.73 AKR1C3 (0.33) SMN1; SMN2ALDH1A1HPGDLMNA
SCHEMBL22499953 0.73 KDM4E (0.32) KMT2A
SCHEMBL27953254 0.73 SLC6A2 (0.43) SMN1; SMN2GABRDGABRA1GABRB1GABRA5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1776357-A1 HYDROXYAMIDE COMPOUNDS HAVING ACTIVITY AS INHIBITORS OF HISTONE DEACETYLASE (HDAC) Astellas Pharma Inc. (JP) 2007-04-25 EP disclosed
WO-2006016680-A1 HYDROXYAMIDE COMPOUNDS HAVING ACTIVITY AS INHIBITORS OF HISTONE DEACETYLASE (HDAC) ASTELLAS PHARMA INC. (JP) 2006-02-16 WO disclosed