SCHEMBL5169133

SCHEMBL5169133

O=C(O)/C=C/c1cnc(N[C@@]2(Cc3cccc(Cl)c3)CCCNC2)cn1

nearest known ligand 0.44

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.35
TAAR1 Q96RJ0 1/20 0.35
SSTR1 P30872 1/20 0.35
SSTR4 P31391 1/20 0.35
HCAR2 Q8TDS4 1/20 0.34
HPGD P15428 1/20 0.32
HSD11B1 P28845 1/20 0.32
CA2 P00918 1/20 0.32
CA5A P35218 1/20 0.32
CA9 Q16790 1/20 0.32
GAA P10253 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5197780 0.90 HDAC3 (0.38) ALDH1A1
SCHEMBL5171832 0.89 RAB9A (0.31) ALDH1A1TAAR1
SCHEMBL5197786 0.85 SLC6A2 (0.36) ALDH1A1SSTR1SSTR4CA2CA5A
SCHEMBL5197021 0.85 AKR1C3 (0.34) ALDH1A1
SCHEMBL5191421 0.84 HDAC3 (0.39) ALDH1A1HCAR2
SCHEMBL5171686 0.84 SLC6A2 (0.35) HCAR2CA2CA5ACA9
SCHEMBL5169616 0.84 MAPKAPK2 (0.31) ALDH1A1
SCHEMBL5167688 0.84 AKR1C3 (0.32) ALDH1A1
SCHEMBL5195227 0.83 RAB9A (0.32) TAAR1CA2CA5ACA9GAA
SCHEMBL5170203 0.83 SLC6A2 (0.38)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1776357-A1 HYDROXYAMIDE COMPOUNDS HAVING ACTIVITY AS INHIBITORS OF HISTONE DEACETYLASE (HDAC) Astellas Pharma Inc. (JP) 2007-04-25 EP disclosed
WO-2006016680-A1 HYDROXYAMIDE COMPOUNDS HAVING ACTIVITY AS INHIBITORS OF HISTONE DEACETYLASE (HDAC) ASTELLAS PHARMA INC. (JP) 2006-02-16 WO disclosed