SCHEMBL5173231

SCHEMBL5173231

NC(=O)c1ccccc1CCCC([O])=O

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.42
MAPT P10636 2/20 0.42
KDM4E B2RXH2 2/20 0.42
HPGD P15428 1/20 0.42
TSHR P16473 1/20 0.42
HSD17B10 Q99714 1/20 0.42
FOLH1 Q04609 1/20 0.41
METAP2 P50579 1/20 0.40
LMNA P02545 2/20 0.39
BCAT2 O15382 1/20 0.39
KMT2A Q03164 3/20 0.38
MEN1 O00255 2/20 0.38
SLC6A3 Q01959 2/20 0.37
HDAC6 Q9UBN7 2/20 0.37
NR1I2 O75469 1/20 0.37
CHRM2 P08172 1/20 0.37
CYP3A4 P08684 1/20 0.37
ADRA2A P08913 1/20 0.37
OPRK1 P41145 1/20 0.37
HTR2B P41595 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5157746 0.89 ALDH1A1 (0.45) ALDH1A1MAPTKDM4EHPGDTSHR
SCHEMBL30177551 0.87 ALDH1A1 (0.50) ALDH1A1MAPTKDM4EHPGDTSHR
SCHEMBL31054164 0.85 MAPT (0.48) ALDH1A1MAPTKDM4EHPGDTSHR
SCHEMBL4735612 0.82 ALDH1A1 (0.54) ALDH1A1MAPTKDM4EHPGDTSHR
SCHEMBL3262902 0.81 ALDH1A1 (0.45) ALDH1A1MAPTKDM4EHPGDTSHR
SCHEMBL2021481 0.81 BCAT2 (0.46) ALDH1A1MAPTKDM4EHPGDTSHR
SCHEMBL3379979 0.80 BCAT2 (0.44) ALDH1A1MAPTKDM4EHPGDTSHR
SCHEMBL30839543 0.80 ALDH1A1 (0.44) ALDH1A1MAPTKDM4EHPGDTSHR
SCHEMBL1002853 0.80 MAPT (0.53) ALDH1A1MAPTKDM4EHPGDTSHR
Bromide SCHEMBL4760758 0.79 MAPT (0.51) ALDH1A1MAPTKDM4EHPGDTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1745022-B1 HISTONE DEACETYLASE INHIBITOR PRODRUGS ATON PHARMA INC (US) 2014-08-13 EP claimed
US-8227636-B2 Histone deacetylase inhibitor prodrugs MERCK HDAC RESEARCH, LLC (US) 2012-07-24 US claimed
EP-1745022-B1 HISTONE DEACETYLASE INHIBITOR PRODRUGS ATON PHARMA INC (US) 2014-08-13 EP disclosed
EP-1745022-A1 HISTONE DEACETYLASE INHIBITOR PRODRUGS Aton Pharma, Inc. (US) 2007-01-24 EP disclosed
WO-2005097747-A1 HISTONE DEACETYLASE INHIBITOR PRODRUGS ATON PHARMA, INC. (US) 2005-10-20 WO disclosed