SCHEMBL5157746

SCHEMBL5157746

NC(=O)c1ccccc1CCC([O])=O

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.45
KDM4E B2RXH2 2/20 0.45
MAPT P10636 1/20 0.45
HPGD P15428 1/20 0.45
TSHR P16473 1/20 0.45
HSD17B10 Q99714 1/20 0.45
LMNA P02545 1/20 0.45
FOLH1 Q04609 1/20 0.43
METAP2 P50579 1/20 0.42
BCAT2 O15382 1/20 0.41
KMT2A Q03164 2/20 0.40
MEN1 O00255 1/20 0.40
SIRT2 Q8IXJ6 1/20 0.38
GAA P10253 1/20 0.38
CTNNB1 P35222 1/20 0.38
SIRT1 Q96EB6 1/20 0.38
MAPK8 P45983 1/20 0.37
IRAK4 Q9NWZ3 1/20 0.37
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5173231 0.89 ALDH1A1 (0.42) ALDH1A1KDM4EMAPTHPGDTSHR
SCHEMBL4735612 0.86 ALDH1A1 (0.54) ALDH1A1KDM4EMAPTHPGDTSHR
SCHEMBL17871919 0.85 KEAP1 (0.50) ALDH1A1KDM4EMAPTHPGDTSHR
SCHEMBL6365140 0.83 ALDH1A1 (0.65) ALDH1A1KDM4EMAPTHPGDTSHR
SCHEMBL27568253 0.82 FOLH1 (0.63) ALDH1A1KDM4EMAPTHPGDTSHR
SCHEMBL30177551 0.82 ALDH1A1 (0.50) ALDH1A1KDM4EMAPTHPGDTSHR
SCHEMBL31054164 0.80 MAPT (0.48) ALDH1A1KDM4EMAPTHPGDTSHR
SCHEMBL731621 0.80 HMGB1 (0.55) ALDH1A1KDM4EMAPTHPGDTSHR
SCHEMBL363595 0.80 BCAT2 (0.48) ALDH1A1KDM4EMAPTHPGDTSHR
SCHEMBL27576949 0.80 ALDH1A1 (0.48) ALDH1A1KDM4EMAPTHPGDTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1745022-B1 HISTONE DEACETYLASE INHIBITOR PRODRUGS ATON PHARMA INC (US) 2014-08-13 EP claimed
US-8227636-B2 Histone deacetylase inhibitor prodrugs MERCK HDAC RESEARCH, LLC (US) 2012-07-24 US claimed
EP-1745022-B1 HISTONE DEACETYLASE INHIBITOR PRODRUGS ATON PHARMA INC (US) 2014-08-13 EP disclosed
EP-1745022-A1 HISTONE DEACETYLASE INHIBITOR PRODRUGS Aton Pharma, Inc. (US) 2007-01-24 EP disclosed
WO-2005097747-A1 HISTONE DEACETYLASE INHIBITOR PRODRUGS ATON PHARMA, INC. (US) 2005-10-20 WO disclosed