SCHEMBL5178358

SCHEMBL5178358

[CH2][C@](O)(c1ccc(Cl)nc1)C(C)(C)C

nearest known ligand 0.37

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.37
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
NAPRT Q6XQN6 1/20 0.36
KCNQ3 O43525 4/20 0.36
KCNQ2 O43526 4/20 0.36
KCNE1 P15382 3/20 0.36
KCNQ1 P51787 3/20 0.36
ADRA2A P08913 2/20 0.34
ADRA2B P18089 2/20 0.34
ADRA2C P18825 2/20 0.34
DGAT1 O75907 2/20 0.34
GRM4 Q14833 1/20 0.33
GAA P10253 1/20 0.33
PIK3CD O00329 1/20 0.32
RAB9A P51151 1/20 0.32
BACE1 P56817 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29978443 0.80 MEN1 (0.41) ALDH1A1MEN1KMT2ANAPRTKCNQ3
SCHEMBL248240 0.80 MEN1 (0.41) ALDH1A1MEN1KMT2ANAPRTKCNQ3
SCHEMBL27311270 0.80 ALDH1A1 (0.37) ALDH1A1NAPRTKCNQ3KCNQ2KCNE1
SCHEMBL29909266 0.76 POLB (0.40) ALDH1A1NAPRTKCNQ3KCNQ2KCNE1
SCHEMBL77078 0.76 POLB (0.40) ALDH1A1NAPRTKCNQ3KCNQ2KCNE1
SCHEMBL31000265 0.74 GCK (0.46) KCNQ3KCNQ2KCNE1KCNQ1GRM4
SCHEMBL18053748 0.74 GCK (0.46) KCNQ3KCNQ2KCNE1KCNQ1GRM4
SCHEMBL31000262 0.74 GCK (0.46) KCNQ3KCNQ2KCNE1KCNQ1GRM4
SCHEMBL12925545 0.73 DGAT1 (0.40) ALDH1A1DGAT1GAARAB9A
SCHEMBL24746455 0.73 MAPT (0.41) ALDH1A1MEN1KMT2ANAPRTKCNQ3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1791811-A1 AMINOALCOHOL DERIVATIVES Astellas Pharma Inc. (JP) 2007-06-06 EP disclosed
EP-1697301-A2 AMINOALCOHOL DERIVATIVES Astellas Pharma Inc. (JP) 2006-09-06 EP disclosed
WO-2006033446-A1 AMINOALCOHOL DERIVATIVES ASTELLAS PHARMA INC. (JP) 2006-03-30 WO disclosed
WO-2005061433-A2 AMINOALCOHOL DERIVATIVES ASTELLAS PHARMA INC. (JP) 2005-07-07 WO disclosed