SCHEMBL5183256

SCHEMBL5183256

[c]1ccccc1-c1cocn1

nearest known ligand 0.37

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 2/20 0.37
HDAC4 P56524 1/20 0.36
KCNK13 Q9HB14 1/20 0.35
FAAH O00519 1/20 0.33
EDNRB P24530 1/20 0.31
EDNRA P25101 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9199874 0.73 SCN9A (0.33) SCN9AKCNK13
SCHEMBL19584694 0.72 F2RL1 (0.37) SCN9A
SCHEMBL37815 0.71 KDM4E (0.54)
SCHEMBL69569 0.71
SCHEMBL648786 0.70 SCN9A (0.53) SCN9AHDAC4FAAHEDNRBEDNRA
SCHEMBL22388750 0.69 SCN9A (0.37) SCN9AHDAC4KCNK13
SCHEMBL115447 0.69 CYP3A4 (0.33)
SCHEMBL26259957 0.68 SCN9A (0.44) SCN9AHDAC4KCNK13FAAHEDNRB
SCHEMBL467328 0.68 MDM2 (0.35)
SCHEMBL18543166 0.68 SCN9A (0.44) SCN9AHDAC4EDNRBEDNRA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1799637-A1 SUBSTITUTED SULFONAMIDOPROPIONAMIDES AND METHODS OF USE Amgen, Inc (US) 2007-06-27 EP claimed
WO-2006036664-A1 SUBSTITUTED SULFONAMIDOPROPIONAMIDES AND METHODS OF USE AMGEN INC. (US) 2006-04-06 WO claimed
EP-1799637-A1 SUBSTITUTED SULFONAMIDOPROPIONAMIDES AND METHODS OF USE Amgen, Inc (US) 2007-06-27 EP disclosed
WO-2006036664-A1 SUBSTITUTED SULFONAMIDOPROPIONAMIDES AND METHODS OF USE AMGEN INC. (US) 2006-04-06 WO disclosed