SCHEMBL5186198

SCHEMBL5186198

CCCS(=O)(=O)NCC(C)(F)c1ccc(-c2ccc(C(N)=O)cc2)cc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.38
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
CA9 Q16790 1/20 0.38
CA14 Q9ULX7 1/20 0.38
EPHX2 P34913 1/20 0.38
NR1H4 Q96RI1 1/20 0.38
P2RY14 Q15391 3/20 0.37
KIF11 P52732 3/20 0.37
RORC P51449 1/20 0.37
MAP2K4 P45985 2/20 0.37
CCR6 P51684 1/20 0.36
MAOB P27338 1/20 0.34
HSD11B1 P28845 1/20 0.34
TP53 P04637 1/20 0.34
ESRRG P62508 1/20 0.34
ALDH1A1 P00352 1/20 0.33
MAPK1 P28482 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
KDM4E B2RXH2 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5186063 0.89 RXRA (0.40) EPHX2KIF11ALDH1A1
SCHEMBL5187403 0.87 HDAC4 (0.43) CA12CA9EPHX2NR1H4P2RY14
SCHEMBL5186061 0.86 KIF11 (0.36) CA2P2RY14KIF11RORC
SCHEMBL6561643 0.84 ALDH1A1 (0.39) CA12CA1CA2CA9KIF11
SCHEMBL5186197 0.83 KIF11 (0.41) KIF11ALDH1A1SMN1; SMN2
SCHEMBL5186164 0.82 KIF11 (0.50) CA12CA1CA2CA9CA14
SCHEMBL6155949 0.82 KIF11 (0.50) CA12CA1CA2CA9CA14
SCHEMBL6155989 0.82 KIF11 (0.50) CA12CA1CA2CA9CA14
SCHEMBL5186003 0.82 HPGD (0.47) ALDH1A1MAPK1SMN1; SMN2KDM4E
SCHEMBL5186190 0.81 GRIA4 (0.44) CA12CA1CA2CA9CA14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1183232-B1 MONOFLUOROALKYL DERIVATIVES LILLY CO ELI (US) 2007-10-03 EP claimed