SCHEMBL5192115

SCHEMBL5192115

COc1ccc(CCN2CCOC(C(N)=O)C2)cc1OC

nearest known ligand 0.49

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
DRD4 P21917 1/20 0.48
SIGMAR1 Q99720 3/20 0.48
EBP Q15125 2/20 0.48
TMEM97 Q5BJF2 1/20 0.48
CHRM3 P20309 1/20 0.48
MEN1 O00255 1/20 0.47
KMT2A Q03164 1/20 0.47
DHCR7 Q9UBM7 1/20 0.47
LMNA P02545 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
HTT P42858 1/20 0.46
POLB P06746 1/20 0.46
ALDH1A1 P00352 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5194021 0.86 SIGMAR1 (0.54) DRD4SIGMAR1
SCHEMBL5378298 0.79 DRD4 (0.47) DRD4SIGMAR1MEN1KMT2APOLB
SCHEMBL5196325 0.76 DRD4 (0.64) DRD4SMN1; SMN2
SCHEMBL8828288 0.75 SIGMAR1 (0.54) SIGMAR1EBPTMEM97DHCR7
SCHEMBL3552685 0.75 SIGMAR1 (0.49) SIGMAR1EBPTMEM97CHRM3ALDH1A1
SCHEMBL3560527 0.75 SIGMAR1 (0.49) SIGMAR1EBPTMEM97CHRM3ALDH1A1
SCHEMBL10511464 0.74 EBP (0.56) SIGMAR1EBPTMEM97DHCR7LMNA
SCHEMBL27334030 0.74 SIGMAR1 (0.56) SIGMAR1EBPTMEM97CHRM3MEN1
SCHEMBL9739025 0.73 HTR1A (0.56) SIGMAR1EBPTMEM97DHCR7
SCHEMBL7351513 0.73 SIGMAR1 (0.53) SIGMAR1EBPTMEM97CHRM3MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0968206-B8 N-HETEROCYCLIC DERIVATIVES AS NOS INHIBITORS BERLEX INC (US) 2007-01-24 EP claimed
EP-0968206-A1 N-HETEROCYCLIC DERIVATIVES AS NOS INHIBITORS BERLEX LABORATORIES, INC. (US) 2000-01-05 EP claimed
WO-1998037079-A1 N-HETEROCYCLIC DERIVATIVES AS NOS INHIBITORS BERLEX LABORATORIES, INC. (US) 1998-08-27 WO claimed