SCHEMBL5194162

SCHEMBL5194162

FC(F)(F)c1ccc(-c2ccccc2-c2ccc(C(F)(F)F)cc2)cc1.Fc1ccc(I)c(Br)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NTRK1 P04629 1/20 0.41
KIF11 P52732 1/20 0.41
PIK3R1 P27986 1/20 0.37
PIK3CA P42336 1/20 0.37
BACE1 P56817 2/20 0.36
PTGS1 P23219 1/20 0.36
PTGS2 P35354 1/20 0.36
MAOB P27338 1/20 0.36
ENPP1 P22413 1/20 0.36
TOP1 P11387 3/20 0.36
KDM4E B2RXH2 2/20 0.35
NPSR1 Q6W5P4 1/20 0.35
PSEN1 P49768 1/20 0.35
PSEN2 P49810 1/20 0.35
APH1B Q8WW43 1/20 0.35
NCSTN Q92542 1/20 0.35
APH1A Q96BI3 1/20 0.35
PSENEN Q9NZ42 1/20 0.35
ALDH1A1 P00352 1/20 0.34
CYP1A2 P05177 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17840160 0.75 KIF11 (0.68) KIF11BACE1MAOBTOP1KDM4E
SCHEMBL1345566 0.75
SCHEMBL30759017 0.75
SCHEMBL18587184 0.74 NTRK1 (0.46) NTRK1KIF11TOP1APPCLK1
SCHEMBL4597238 0.73 PSEN1 (0.51) KIF11PSEN1PSEN2APH1BNCSTN
SCHEMBL2841464 0.73 ALDH1A1 (0.58) KIF11PIK3R1PIK3CABACE1MAOB
SCHEMBL30053194 0.73 ALDH1A1 (0.58) KIF11PIK3R1PIK3CABACE1MAOB
SCHEMBL5695818 0.73 KIF11 (0.56) NTRK1KIF11BACE1MAOBTOP1
SCHEMBL30116692 0.73 PTPN5 (0.38) KIF11BACE1KDM4ENPSR1ALDH1A1
SCHEMBL3544291 0.73 PTPN5 (0.38) KIF11BACE1KDM4ENPSR1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1773315-A1 ARYLACETIC ACIDS AND RELATED COMPOUNDS FOR TREATMENT OF ALZHEIMER'S DISEASE Merck Sharp & Dohme Limited (GB) 2007-04-18 EP disclosed
WO-2006008558-A1 ARYLACETIC ACIDS AND RELATED COMPOUNDS FOR TREATMENT OF ALZHEIMER’S DISEASE MERCK SHARP & DOHME LIMITED (GB) 2006-01-26 WO disclosed