SCHEMBL5196158

SCHEMBL5196158

CCC(CC)c1nc(-c2ccncc2)c(-c2ccc(Cl)cc2)n1CC.O=C(C(=NO)c1ccncc1)c1ccc(Cl)cc1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LSS P48449 1/20 0.34
BRAF P15056 1/20 0.33
MAPK3 P27361 1/20 0.33
MAPK1 P28482 1/20 0.33
CNR1 P21554 5/20 0.32
GRM1 Q13255 1/20 0.32
CSNK1D P48730 1/20 0.32
CSNK1E P49674 1/20 0.32
MAPK14 Q16539 4/20 0.32
MAPK11 Q15759 2/20 0.32
ROCK2 O75116 1/20 0.32
PRKACA P17612 1/20 0.32
RPS6KB1 P23443 1/20 0.32
IRAK1 P51617 1/20 0.32
PRKX P51817 1/20 0.32
LIMK1 P53667 1/20 0.32
PRKG2 Q13237 1/20 0.32
ROCK1 Q13464 1/20 0.32
PRKG1 Q13976 1/20 0.32
PKN2 Q16513 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5200281 0.93 LSS (0.33) LSSBRAFMAPK3MAPK1CNR1
SCHEMBL5330737 0.90 CNR1 (0.39) LSSBRAFMAPK3MAPK1CNR1
SCHEMBL5200392 0.84 MAPK14 (0.41) LSSMAPK14MAPK11MAPK13MAPK12
SCHEMBL5197704 0.81 KMT2A (0.48) ALDH1A1NPSR1TEK
SCHEMBL5197710 0.81 KMT2A (0.48) ALDH1A1NPSR1TEK
SCHEMBL5199263 0.78 NPC1 (0.37) BRAFCSNK1DCSNK1EMAPK14MAPK11
SCHEMBL5199254 0.78 NPC1 (0.37) BRAFCSNK1DCSNK1EMAPK14MAPK11
SCHEMBL5199937 0.76 MAPK14 (0.42) LSSCNR1MAPK14MAPK11MAPK13
SCHEMBL5198449 0.75 AAK1 (0.42) LSSCNR1MAPK14MAPK11MAPK13
SCHEMBL5197840 0.74 MAOB (0.37) LSSMAPK1MAPK14MAPK11NPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1846389-A1 IMIDAZOLE DERIVATIVES F. Hoffmann-Roche AG (CH) 2007-10-24 EP disclosed
WO-2006082002-A1 IMIDAZOLE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2006-08-10 WO disclosed