SCHEMBL5197178

SCHEMBL5197178

CC(=CCC(C)NC(=O)OC(C)(C)C)c1cncc(Br)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2C19 P33261 1/20 0.41
KDM4E B2RXH2 2/20 0.39
CASP3 P42574 2/20 0.39
AAK1 Q2M2I8 6/20 0.39
ALDH1A1 P00352 4/20 0.38
MAPT P10636 3/20 0.38
MEN1 O00255 3/20 0.38
KMT2A Q03164 3/20 0.38
MAPK1 P28482 3/20 0.38
LMNA P02545 2/20 0.38
GAA P10253 2/20 0.38
TP53 P04637 2/20 0.38
HPGD P15428 1/20 0.38
USP2 O75604 1/20 0.37
ALOX15 P16050 1/20 0.37
POLB P06746 1/20 0.37
HCAR2 Q8TDS4 1/20 0.37
TAS1R3 Q7RTX0 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6462042 0.86 ACACB (0.35) AAK1ALDH1A1MAPTMEN1KMT2A
SCHEMBL3910420 0.85 CHRNB2 (0.38) KDM4EAAK1MAPTKMT2ALMNA
SCHEMBL5224591 0.77 CDK8 (0.39) AAK1
SCHEMBL5197286 0.75 CA1 (0.35) AAK1MAPTLMNA
SCHEMBL6451903 0.75 NNMT (0.41) KDM4EAAK1MAPTMEN1KMT2A
SCHEMBL6853669 0.74 AAK1 (0.43) CYP1A2CYP3A4CYP2C19AAK1
SCHEMBL6853676 0.74 AAK1 (0.43) CYP1A2CYP3A4CYP2C19AAK1
SCHEMBL6453865 0.73 KDM4E (0.44) CYP1A2CYP3A4CYP2C19KDM4ECASP3
SCHEMBL31226247 0.72 KMT2A (0.44) CYP1A2CYP3A4CYP2C19AAK1ALDH1A1
SCHEMBL31226229 0.72 CYP1A2 (0.41) CYP1A2CYP3A4CYP2C19KDM4ECASP3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1814852-A2 HYDROXYBENZOATE SALTS OF METANICOTINE COMPOUNDS Targacept, Inc. (US) 2007-08-08 EP disclosed
EP-1814853-A2 HYDROXYBENZOATE SALTS OF METANICOTINE COMPOUNDS Targacept, Inc. (US) 2007-08-08 EP disclosed
WO-2006053082-A2 HYDROXYBENZOATE SALTS OF METANICOTINE COMPOUNDS TARGACEPT, INC. (US) 2006-05-18 WO disclosed
WO-2006053039-A2 HYDROXYBENZOATE SALTS OF METANICOTINE COMPOUNDS TARGACEPT, INC. (US) 2006-05-18 WO disclosed