SCHEMBL5199512

SCHEMBL5199512

CCOC(=O)CCC(N)c1cc(C)nc(-c2ncc[nH]2)n1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.35
KDM4E B2RXH2 3/20 0.33
ALDH1A1 P00352 3/20 0.33
L3MBTL1 Q9Y468 2/20 0.32
HSD17B10 Q99714 2/20 0.32
ABL1 P00519 1/20 0.32
PKM P14618 1/20 0.32
RIN1 Q13671 1/20 0.32
HPGD P15428 1/20 0.32
MAPT P10636 2/20 0.32
GAA P10253 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31
SYK P43405 1/20 0.31
HCRTR1 O43613 1/20 0.31
HCRTR2 O43614 1/20 0.31
PDE3B Q13370 1/20 0.31
PDE3A Q14432 1/20 0.31
P2RY12 Q9H244 1/20 0.31
HSF1 Q00613 1/20 0.31
POLB P06746 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5202337 0.83 KDM4E (0.36) TSHRKDM4EALDH1A1GAANPSR1
SCHEMBL3559045 0.70 ALDH1A1 (0.41) TSHRKDM4EALDH1A1ABL1RIN1
SCHEMBL5199693 0.67 MAPT (0.34) TSHRKDM4EALDH1A1HSD17B10PKM
SCHEMBL11826761 0.65 ALDH1A1 (0.57) KDM4EALDH1A1HPGDMAPTKMT2A
SCHEMBL5204329 0.64 KDM4E (0.39) KDM4EALDH1A1SYKHCRTR1HCRTR2
SCHEMBL3507805 0.64 ALDH1A1 (0.54) KDM4EALDH1A1KMT2A
SCHEMBL8537268 0.63 SYK (0.51) KDM4EALDH1A1HSD17B10MAPTSYK
SCHEMBL5200407 0.63 KDM4E (0.41) KDM4EALDH1A1
SCHEMBL3591993 0.63 MAPT (0.52) KDM4EALDH1A1L3MBTL1HSD17B10MAPT
SCHEMBL5200333 0.62 KDM4E (0.39) KDM4EALDH1A1MAPTHCRTR1HCRTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1817030-A2 INDUCIBLE NITRIC OXIDE SYNTHASE DIMERIZATION INHIBITORS Kalypsys, Inc. (US) 2007-08-15 EP disclosed
WO-2006060424-A2 INDUCIBLE NITRIC OXIDE SYNTHASE DIMERIZATION INHIBITORS KALYPSYS, INC. (US) 2006-06-08 WO disclosed