SCHEMBL5202337

SCHEMBL5202337

CCOC(=O)C(N)c1cc(C)nc(-c2ncc[nH]2)n1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.36
ALDH1A1 P00352 2/20 0.36
HSF1 Q00613 2/20 0.35
GAA P10253 2/20 0.34
HTT P42858 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
MAPK14 Q16539 1/20 0.32
GRIA1 P42261 1/20 0.32
GRIA2 P42262 1/20 0.32
GRIA3 P42263 1/20 0.32
GRIA4 P48058 1/20 0.32
PDE4A P27815 2/20 0.32
PDE4B Q07343 2/20 0.32
PDE4C Q08493 2/20 0.32
PDE4D Q08499 2/20 0.32
PKN1 Q16512 1/20 0.32
PKN2 Q16513 1/20 0.32
SMPD3 Q9NY59 1/20 0.32
HCRTR1 O43613 1/20 0.31
HCRTR2 O43614 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5199512 0.83 TSHR (0.35) KDM4EALDH1A1HSF1GAANPSR1
SCHEMBL5199693 0.71 MAPT (0.34) KDM4EALDH1A1HSF1NPSR1MAPK14
SCHEMBL5204329 0.68 KDM4E (0.39) KDM4EALDH1A1HSF1MAPK14PDE4A
SCHEMBL3507805 0.67 ALDH1A1 (0.54) KDM4EALDH1A1PDE4APDE4BPDE4C
SCHEMBL3560003 0.67 TSHR (0.43) KDM4EALDH1A1HTTMEN1KMT2A
SCHEMBL5200407 0.67 KDM4E (0.41) KDM4EALDH1A1MAPK14SMPD3F10
SCHEMBL5200333 0.66 KDM4E (0.39) KDM4EALDH1A1HSF1MAPK14PDE4A
SCHEMBL5199466 0.66 LMNA (0.46) KDM4EALDH1A1HSF1HTTSMPD3
SCHEMBL5200449 0.65 BRD4 (0.37) KDM4EALDH1A1HSF1PDE4APDE4B
SCHEMBL6171373 0.65 ALDH1A1 (0.42) KDM4EALDH1A1GAAMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1817030-A2 INDUCIBLE NITRIC OXIDE SYNTHASE DIMERIZATION INHIBITORS Kalypsys, Inc. (US) 2007-08-15 EP disclosed
WO-2006060424-A2 INDUCIBLE NITRIC OXIDE SYNTHASE DIMERIZATION INHIBITORS KALYPSYS, INC. (US) 2006-06-08 WO disclosed