SCHEMBL5204329

SCHEMBL5204329

Cc1cc(C(C)(C)C(N)=O)nc(-c2ncc[nH]2)n1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.39
ALDH1A1 P00352 2/20 0.39
CSNK1A1 P48729 2/20 0.36
TYRO3 Q06418 1/20 0.36
DYRK1B Q9Y463 1/20 0.36
PDE4A P27815 2/20 0.36
PDE4B Q07343 2/20 0.36
PDE4C Q08493 2/20 0.36
PDE4D Q08499 2/20 0.36
NISCH Q9Y2I1 1/20 0.36
HCRTR1 O43613 1/20 0.35
HCRTR2 O43614 1/20 0.35
PARP1 P09874 1/20 0.34
MAPK14 Q16539 2/20 0.34
SMPD3 Q9NY59 1/20 0.34
SYK P43405 1/20 0.32
TRPV1 Q8NER1 1/20 0.32
BRD4 O60885 1/20 0.32
NPC1 O15118 1/20 0.32
RAB9A P51151 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5200333 0.88 KDM4E (0.39) KDM4EALDH1A1CSNK1A1TYRO3DYRK1B
SCHEMBL5200348 0.78 NISCH (0.34) ALDH1A1NISCHHCRTR1HCRTR2SMPD3
SCHEMBL5199466 0.69 LMNA (0.46) KDM4EALDH1A1NISCHSMPD3BRD4
SCHEMBL5202337 0.68 KDM4E (0.36) KDM4EALDH1A1PDE4APDE4BPDE4C
SCHEMBL8283628 0.67 CYP19A1 (0.39) KDM4EALDH1A1CSNK1A1TYRO3DYRK1B
SCHEMBL5201640 0.66 KDM4E (0.31) KDM4EALDH1A1
SCHEMBL5200449 0.66 BRD4 (0.37) KDM4EALDH1A1PDE4APDE4BPDE4C
SCHEMBL5200407 0.65 KDM4E (0.41) KDM4EALDH1A1MAPK14SMPD3SMO
SCHEMBL9026316 0.65 NISCH (0.50) KDM4EALDH1A1CSNK1A1TYRO3DYRK1B
SCHEMBL23772037 0.63 NISCH (0.44) KDM4EALDH1A1PDE4APDE4BPDE4C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1817030-A2 INDUCIBLE NITRIC OXIDE SYNTHASE DIMERIZATION INHIBITORS Kalypsys, Inc. (US) 2007-08-15 EP disclosed
WO-2006060424-A2 INDUCIBLE NITRIC OXIDE SYNTHASE DIMERIZATION INHIBITORS KALYPSYS, INC. (US) 2006-06-08 WO disclosed