SCHEMBL5199602

SCHEMBL5199602

Cc1cccc(-c2n[nH]cc2-c2ccc(F)c(-c3ccc(S(N)(=O)=O)c(OC(F)(F)F)c3)c2)n1

nearest known ligand 0.36

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 7/20 0.36
TGFBR1 P36897 4/20 0.36
TRPV1 Q8NER1 2/20 0.33
ALOX5AP P20292 1/20 0.33
FEN1 P39748 1/20 0.33
GHSR Q92847 1/20 0.32
GRM2 Q14416 1/20 0.32
PTGS2 P35354 2/20 0.32
LRRK2 Q5S007 1/20 0.31
PTGS1 P23219 1/20 0.31
PDE3B Q13370 1/20 0.31
PDE3A Q14432 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5198270 0.88 TGFBR1 (0.42) TGFBR1ALOX5APFEN1GHSRPTGS2
SCHEMBL5198316 0.88 TGFBR1 (0.37) TGFBR1ALOX5APFEN1GHSRPTGS2
SCHEMBL5200774 0.87 TGFBR1 (0.39) TGFBR1ALOX5APFEN1GHSRPTGS2
SCHEMBL5199511 0.85 TGFBR1 (0.38) TGFBR1ALOX5APFEN1PTGS2LRRK2
SCHEMBL5198993 0.85 TGFBR1 (0.37) TGFBR1ALOX5APFEN1GHSRPTGS2
SCHEMBL5200017 0.84 TGFBR1 (0.39) TGFBR1ALOX5APFEN1PTGS2LRRK2
SCHEMBL5199208 0.83 TGFBR1 (0.39) TGFBR1ALOX5APFEN1GHSRPTGS2
SCHEMBL5198372 0.83 PTGS2 (0.45) TGFBR1PTGS2LRRK2PTGS1
SCHEMBL5199630 0.80 TGFBR1 (0.42) TGFBR1PTGS2
SCHEMBL5199341 0.78 TGFBR1 (0.44) TGFBR1PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20070275968-A1 Substituted Biphenyl Derivative SANKYO COMPANY, LIMITED (JP) 2007-11-29 US disclosed
EP-1798229-A1 SUBSTITUTED BIPHENYL DERIVATIVE Sankyo Company, Limited (JP) 2007-06-20 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070275968-A1 Substituted Biphenyl Derivative COL2A1, COL1A1, FGFR3 SCN9A 4074/4885TGFBR1 40/4885TRPV1 2364/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.