SCHEMBL5200348

SCHEMBL5200348

Cc1cc(C(C)(C)CN)nc(-c2ncc[nH]2)n1

nearest known ligand 0.34

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
NISCH Q9Y2I1 1/20 0.34
HSF1 Q00613 2/20 0.32
BRD4 O60885 1/20 0.31
ADORA2A P29274 1/20 0.30
ADORA1 P30542 1/20 0.30
HCRTR1 O43613 1/20 0.30
HCRTR2 O43614 1/20 0.30
ALDH1A1 P00352 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30
SMPD3 Q9NY59 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5204329 0.78 KDM4E (0.39) NISCHHSF1BRD4HCRTR1HCRTR2
SCHEMBL5200333 0.77 KDM4E (0.39) NISCHHSF1BRD4HCRTR1HCRTR2
SCHEMBL5199466 0.71 LMNA (0.46) NISCHHSF1BRD4ADORA2AADORA1
SCHEMBL5200449 0.68 BRD4 (0.37) NISCHHSF1BRD4ADORA2AADORA1
SCHEMBL9026316 0.67 NISCH (0.50) NISCHHSF1BRD4ALDH1A1SMN1; SMN2
SCHEMBL23772037 0.65 NISCH (0.44) NISCHHSF1ADORA2AADORA1ALDH1A1
SCHEMBL5202337 0.64 KDM4E (0.36) HSF1HCRTR1HCRTR2ALDH1A1SMN1; SMN2
SCHEMBL4554721 0.63 NISCH (0.42) NISCHHSF1ADORA2AADORA1ALDH1A1
SCHEMBL10721690 0.62 SMN1; SMN2 (0.41) NISCHALDH1A1SMN1; SMN2
SCHEMBL5200407 0.62 KDM4E (0.41) ADORA2AADORA1ALDH1A1SMPD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1817030-A2 INDUCIBLE NITRIC OXIDE SYNTHASE DIMERIZATION INHIBITORS Kalypsys, Inc. (US) 2007-08-15 EP disclosed
WO-2006060424-A2 INDUCIBLE NITRIC OXIDE SYNTHASE DIMERIZATION INHIBITORS KALYPSYS, INC. (US) 2006-06-08 WO disclosed