SCHEMBL5200482

SCHEMBL5200482

CCN(CC)C(=O)Oc1ccc2c(N)cccc2n1

nearest known ligand 0.49

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TSPO P30536 6/20 0.49
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
LMNA P02545 4/20 0.40
SMN1; SMN2 Q16637 3/20 0.40
NPC1 O15118 2/20 0.40
RAB9A P51151 2/20 0.40
MAPT P10636 1/20 0.40
KDM4E B2RXH2 2/20 0.40
L3MBTL1 Q9Y468 2/20 0.39
TSHR P16473 1/20 0.39
ALDH1A1 P00352 1/20 0.38
NFKB1 P19838 1/20 0.38
NFKB2 Q00653 1/20 0.38
RELA Q04206 1/20 0.38
HSD17B10 Q99714 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5203518 0.79 KMT2A (0.41) MEN1KMT2ALMNANPC1RAB9A
SCHEMBL5206188 0.78 HTR3A (0.40) MEN1KMT2ALMNANPC1RAB9A
SCHEMBL4820741 0.77 KDM4A (0.50) MEN1KMT2ALMNASMN1; SMN2NPC1
SCHEMBL5201133 0.77 ALDH1A1 (0.43) KMT2ALMNANPC1RAB9AMAPT
SCHEMBL7812110 0.74 HTR3A (0.36) KMT2ALMNANPC1RAB9AKDM4E
SCHEMBL4816736 0.74 ALDH1A1 (0.46) KMT2ALMNANPC1RAB9AKDM4E
SCHEMBL10675880 0.73 TSPO (0.60) TSPOMEN1KMT2ASMN1; SMN2NPC1
SCHEMBL3532637 0.72 HTR3A (0.46) MEN1KMT2ALMNANPC1RAB9A
SCHEMBL31179390 0.72 HTR3A (0.46) MEN1KMT2ALMNANPC1RAB9A
SCHEMBL9326908 0.72 MEN1 (0.50) TSPOMEN1KMT2ALMNASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1492771-B1 QUINOLINE AND ISOQUINOLINE DERIVATIVES, METHOD FOR THE PRODUCTION THEREOF AND USE THEREOF AS ANTI-INFLAMMATORY AGENTS SCHERING AG (DE) 2007-02-28 EP disclosed
EP-1492771-A1 QUINOLINE AND ISOQUINOLINE DERIVATIVES, METHOD FOR THE PRODUCTION THEREOF AND USE THEREOF AS ANTI-INFLAMMATORY AGENTS SCHERING AKTIENGESELLSCHAFT (DE) 2005-01-05 EP disclosed
WO-2003082827-A1 QUINOLINE AND ISOQUINOLINE DERIVATIVES, METHOD FOR THE PRODUCTION THEREOF AND USE THEREOF AS ANTI-INFLAMMATORY AGENTS SCHERING AKTIENGESELLSCHAFT (DE) 2003-10-09 WO disclosed