SCHEMBL5201272

SCHEMBL5201272

CN(C)C(=O)Cc1ccc2ccn(C3CCN(CCc4ccccc4F)CC3)c2c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 3/20 0.43
DRD2 P14416 1/20 0.43
SLC6A4 P31645 1/20 0.43
CCR5 P51681 4/20 0.41
HTR2A P28223 1/20 0.40
HTR7 P34969 1/20 0.40
KCNH2 Q12809 1/20 0.40
HTR1A P08908 1/20 0.39
HTR1D P28221 1/20 0.39
HTR1B P28222 1/20 0.39
HTR1F P30939 1/20 0.39
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
OPRD1 P41143 1/20 0.39
OPRK1 P41145 1/20 0.39
CACNA1G O43497 1/20 0.39
CCR4 P51679 1/20 0.38
BLM P54132 1/20 0.38
MCHR1 Q99705 1/20 0.37
CCR3 P51677 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5871014 0.88 CCR5 (0.47) OPRM1CCR5MEN1KMT2ACCR4
SCHEMBL4081913 0.88 DRD2 (0.43) OPRM1DRD2SLC6A4HTR2AHTR7
Oxalic Acid SCHEMBL5871140 0.87 CCR5 (0.49) OPRM1CCR5MEN1KMT2ACCR4
SCHEMBL5871942 0.87 HTR1A (0.48) OPRM1DRD2SLC6A4CCR5HTR2A
SCHEMBL5871701 0.86 DRD2 (0.44) OPRM1DRD2SLC6A4HTR2AHTR7
Oxalic Acid SCHEMBL5871682 0.86 CCR5 (0.47) OPRM1CCR5KCNH2MEN1KMT2A
SCHEMBL5871734 0.85 SLC6A4 (0.46) OPRM1DRD2SLC6A4HTR2AHTR7
Oxalic Acid SCHEMBL5871218 0.85 HTR1A (0.46) OPRM1DRD2SLC6A4CCR5HTR2A
SCHEMBL4076926 0.84 HTR2A (0.44) OPRM1DRD2SLC6A4HTR2AHTR7
SCHEMBL5871274 0.83 CCR3 (0.41) OPRM1DRD2SLC6A4HTR1AHTR1D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1179532-B1 PROCESS FOR THE PRODUCTION OF INDOLE DERIVATIVES AND INTERMEDIATES THEREFOR EISAI R&D MAN CO LTD (JP) 2007-06-13 EP disclosed
US-6573384-B1 1,4-substituted cyclic amine compound which is useful as a pharmaceutical, and an intermediate for the process EISAI CO., LTD. (JP) 2003-06-03 US disclosed
EP-1179532-A1 PROCESS FOR THE PRODUCTION OF INDOLE DERIVATIVES AND INTERMEDIATES THEREFOR Eisai Co., Ltd. (JP) 2002-02-13 EP disclosed