SCHEMBL5201529

SCHEMBL5201529

CCOC(=O)c1csc(C2CCN(C(=O)OC(C)(C)C)C2c2cc(C)nc(-c3ncc[nH]3)n2)n1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR1H2 P55055 1/20 0.43
NR1H3 Q13133 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.35
GAA P10253 1/20 0.34
UCHL1 P09936 2/20 0.34
USP30 Q70CQ3 2/20 0.34
CASP3 P42574 1/20 0.33
CASP7 P55210 1/20 0.33
CASP8 Q14790 1/20 0.33
TPH1 P17752 2/20 0.33
ABCB1 P08183 1/20 0.32
MAPT P10636 2/20 0.32
NPSR1 Q6W5P4 1/20 0.32
HPGD P15428 1/20 0.32
MEN1 O00255 2/20 0.32
KMT2A Q03164 2/20 0.32
ATM Q13315 1/20 0.31
NPC1 O15118 1/20 0.31
ALDH1A1 P00352 1/20 0.31
RAB9A P51151 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5201565 0.85 USP30 (0.36) UCHL1USP30GPR119GRM5
SCHEMBL5202276 0.81 SMN1; SMN2 (0.38) SMN1; SMN2GAACASP3CASP7CASP8
SCHEMBL3572145 0.81 NR1H2 (0.43) NR1H2NR1H3SMN1; SMN2GAAUCHL1
SCHEMBL5203615 0.78 UCHL1 (0.38) UCHL1USP30GPR119GRM5
SCHEMBL5202192 0.77 UCHL1 (0.37) UCHL1USP30GPR119GRM5
SCHEMBL4761317 0.72 NR1H2 (0.46) NR1H2NR1H3SMN1; SMN2GAACASP3
SCHEMBL12789591 0.71 NR1H2 (0.59) NR1H2NR1H3SMN1; SMN2GAACASP3
SCHEMBL8219203 0.71 NR1H2 (0.59) NR1H2NR1H3SMN1; SMN2GAACASP3
SCHEMBL12215951 0.71 NR1H2 (0.59) NR1H2NR1H3SMN1; SMN2GAACASP3
SCHEMBL23975518 0.70 NR1H2 (0.58) NR1H2NR1H3SMN1; SMN2GAACASP3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1817030-A2 INDUCIBLE NITRIC OXIDE SYNTHASE DIMERIZATION INHIBITORS Kalypsys, Inc. (US) 2007-08-15 EP disclosed
WO-2006060424-A2 INDUCIBLE NITRIC OXIDE SYNTHASE DIMERIZATION INHIBITORS KALYPSYS, INC. (US) 2006-06-08 WO disclosed