SCHEMBL5202276

SCHEMBL5202276

CCOC(=O)c1csc(C2CCNC2c2cc(C)nc(-c3ncc[nH]3)n2)n1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 5/20 0.38
CASP3 P42574 1/20 0.37
CASP7 P55210 1/20 0.37
CASP8 Q14790 1/20 0.37
RAB9A P51151 7/20 0.35
NPC1 O15118 6/20 0.35
MAPT P10636 5/20 0.35
ALDH1A1 P00352 3/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
NPSR1 Q6W5P4 2/20 0.33
POLB P06746 2/20 0.33
PKM P14618 1/20 0.33
RXFP1 Q9HBX9 1/20 0.33
LMNA P02545 1/20 0.33
HSD17B10 Q99714 1/20 0.33
HSP90AA1 P07900 3/20 0.33
MAPK1 P28482 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP2C19 P33261 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5201529 0.81 NR1H2 (0.43) SMN1; SMN2CASP3CASP7CASP8RAB9A
SCHEMBL5200864 0.79 ADORA2A (0.33)
SCHEMBL5199693 0.79 MAPT (0.34) MAPTALDH1A1MEN1KMT2ANPSR1
SCHEMBL3558612 0.78 NOS2 (0.37) SMN1; SMN2CASP3CASP7CASP8RAB9A
SCHEMBL3065517 0.70 MAPT (0.54) SMN1; SMN2RAB9ANPC1MAPTALDH1A1
SCHEMBL1228518 0.68 BAZ2A (0.52) SMN1; SMN2CASP3CASP7CASP8RAB9A
SCHEMBL24980831 0.68 CASP3 (0.47) SMN1; SMN2CASP3CASP7CASP8RAB9A
SCHEMBL8219214 0.67 SMN1; SMN2 (0.52) SMN1; SMN2CASP3CASP7CASP8RAB9A
Bromide SCHEMBL5061856 0.67 BAZ2A (0.51) SMN1; SMN2CASP3CASP7CASP8RAB9A
SCHEMBL4641452 0.67 SCN10A (0.35)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1817030-A2 INDUCIBLE NITRIC OXIDE SYNTHASE DIMERIZATION INHIBITORS Kalypsys, Inc. (US) 2007-08-15 EP disclosed
WO-2006060424-A2 INDUCIBLE NITRIC OXIDE SYNTHASE DIMERIZATION INHIBITORS KALYPSYS, INC. (US) 2006-06-08 WO disclosed