SCHEMBL5201542

SCHEMBL5201542

Cc1cc(CN=C(c2ccccc2)c2ccccc2)nc(-c2ncc[nH]2)n1

nearest known ligand 0.39

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
FFAR1 O14842 16/20 0.39
MTOR P42345 1/20 0.37
ADK P55263 1/20 0.37
NISCH Q9Y2I1 1/20 0.37
ALDH1A1 P00352 1/20 0.36
LMNA P02545 1/20 0.36
HTT P42858 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
ADRA2A P08913 1/20 0.36
HCRTR1 O43613 1/20 0.33
HCRTR2 O43614 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5200449 0.70 BRD4 (0.37) FFAR1MTORADKNISCHALDH1A1
SCHEMBL3562250 0.68 NPSR1 (0.46) ALDH1A1LMNAHTTSMN1; SMN2
SCHEMBL5199466 0.66 LMNA (0.46) MTORADKNISCHALDH1A1LMNA
SCHEMBL20840542 0.65 SMN1; SMN2 (0.46) ALDH1A1LMNASMN1; SMN2
SCHEMBL5199947 0.65 HRH3 (0.35) ALDH1A1HTTHCRTR1HCRTR2
SCHEMBL5201190 0.65 MAPK14 (0.33) ALDH1A1HCRTR1HCRTR2
SCHEMBL5200333 0.63 KDM4E (0.39) MTORADKNISCHALDH1A1ADRA2A
SCHEMBL9026316 0.62 NISCH (0.50) MTORADKNISCHALDH1A1SMN1; SMN2
SCHEMBL5200348 0.62 NISCH (0.34) NISCHALDH1A1SMN1; SMN2HCRTR1HCRTR2
SCHEMBL24910869 0.60 NISCH (0.41) MTORADKNISCHALDH1A1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1817030-A2 INDUCIBLE NITRIC OXIDE SYNTHASE DIMERIZATION INHIBITORS Kalypsys, Inc. (US) 2007-08-15 EP disclosed
WO-2006060424-A2 INDUCIBLE NITRIC OXIDE SYNTHASE DIMERIZATION INHIBITORS KALYPSYS, INC. (US) 2006-06-08 WO disclosed