SCHEMBL5201190

SCHEMBL5201190

Cc1cc(CC2NCCC2C(=O)O)nc(-c2ncc[nH]2)n1

nearest known ligand 0.33

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 1/20 0.33
HCRTR1 O43613 1/20 0.32
HCRTR2 O43614 1/20 0.32
KDM4E B2RXH2 2/20 0.32
ALDH1A1 P00352 2/20 0.32
MMP13 P45452 1/20 0.31
ADAM17 P78536 1/20 0.31
FFAR4 Q5NUL3 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5199693 0.73 MAPT (0.34) MAPK14HCRTR1HCRTR2KDM4EALDH1A1
SCHEMBL5199947 0.71 HRH3 (0.35) HCRTR1HCRTR2KDM4EALDH1A1
SCHEMBL5200449 0.68 BRD4 (0.37) HCRTR1HCRTR2KDM4EALDH1A1
SCHEMBL2637675 0.66 SMN1; SMN2 (0.39) HCRTR1HCRTR2KDM4EALDH1A1
SCHEMBL4641452 0.65 SCN10A (0.35) HCRTR1HCRTR2
SCHEMBL5201542 0.65 FFAR1 (0.39) HCRTR1HCRTR2ALDH1A1
SCHEMBL5200333 0.64 KDM4E (0.39) MAPK14HCRTR1HCRTR2KDM4EALDH1A1
SCHEMBL5202000 0.64 MEN1 (0.33) HCRTR1HCRTR2
SCHEMBL5204446 0.64 HCRTR1 (0.37) MAPK14HCRTR1HCRTR2KDM4EALDH1A1
SCHEMBL5202337 0.62 KDM4E (0.36) MAPK14HCRTR1HCRTR2KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1817030-A2 INDUCIBLE NITRIC OXIDE SYNTHASE DIMERIZATION INHIBITORS Kalypsys, Inc. (US) 2007-08-15 EP disclosed
WO-2006060424-A2 INDUCIBLE NITRIC OXIDE SYNTHASE DIMERIZATION INHIBITORS KALYPSYS, INC. (US) 2006-06-08 WO disclosed