SCHEMBL5201609

SCHEMBL5201609

COCNC(=O)c1csc(-c2ncc[nH]2)n1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGDS O60760 1/20 0.42
HPGD P15428 2/20 0.39
CYP1A2 P05177 2/20 0.39
CYP3A4 P08684 2/20 0.39
CYP2C9 P11712 2/20 0.39
CYP2C19 P33261 2/20 0.39
KDM4E B2RXH2 1/20 0.39
ALDH1A1 P00352 1/20 0.39
TLR7 Q9NYK1 5/20 0.38
HDAC1 Q13547 4/20 0.38
HDAC6 Q9UBN7 4/20 0.38
HDAC3 O15379 3/20 0.38
CDC25A P30304 1/20 0.38
CDC25B P30305 1/20 0.38
HDAC8 Q9BY41 1/20 0.36
SLC40A1 Q9NP59 1/20 0.36
MAP3K5 Q99683 1/20 0.36
POLB P06746 2/20 0.35
NPC1 O15118 1/20 0.35
RAB9A P51151 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3065517 0.76 MAPT (0.54) CYP1A2CYP2C19ALDH1A1POLBNPC1
SCHEMBL27609155 0.76 ALDH1A1 (0.46) HPGDSKDM4EALDH1A1TLR7
SCHEMBL7465829 0.76 ALDH1A1 (0.37) HPGDSHPGDCYP1A2CYP3A4CYP2C9
SCHEMBL5200407 0.75 KDM4E (0.41) HPGDSKDM4EALDH1A1
SCHEMBL3062139 0.74 HTR2B (0.48) HPGDSHPGDCYP2C9CYP2C19KDM4E
SCHEMBL722692 0.74 HPGD (0.64) HPGDSHPGDCYP1A2CYP3A4CYP2C9
SCHEMBL7460091 0.74 HPGDS (0.38) HPGDSHPGDKDM4EALDH1A1TLR7
SCHEMBL3569039 0.73 HDAC1 (0.52) HPGDSHPGDCYP1A2CYP3A4CYP2C9
SCHEMBL31216572 0.72 HTR3E (0.37) HPGDCYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL3818165 0.72 MAPT (0.51) HPGDSCYP1A2CYP3A4CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1817030-A2 INDUCIBLE NITRIC OXIDE SYNTHASE DIMERIZATION INHIBITORS Kalypsys, Inc. (US) 2007-08-15 EP disclosed
WO-2006060424-A2 INDUCIBLE NITRIC OXIDE SYNTHASE DIMERIZATION INHIBITORS KALYPSYS, INC. (US) 2006-06-08 WO disclosed