SCHEMBL7460091

SCHEMBL7460091

CC(C)(C)OC(=O)CC(=O)c1csc(-c2ncc[nH]2)n1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGDS O60760 1/20 0.38
KDM4E B2RXH2 1/20 0.35
ALDH1A1 P00352 1/20 0.35
SCN9A Q15858 1/20 0.34
TLR7 Q9NYK1 2/20 0.33
HDAC1 Q13547 4/20 0.32
HDAC6 Q9UBN7 4/20 0.32
HDAC3 O15379 3/20 0.32
ACKR3 P25106 1/20 0.32
HPGD P15428 1/20 0.32
SREBF2 Q12772 1/20 0.32
ABCB1 P08183 1/20 0.32
SMPD3 Q9NY59 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
HDAC8 Q9BY41 1/20 0.30
CDC25A P30304 1/20 0.30
CDC25B P30305 1/20 0.30
CCNB2 O95067 1/20 0.30
CCNE2 O96020 1/20 0.30
CDK1 P06493 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7707033 0.81 HPGDS (0.38) HPGDSALDH1A1HDAC1HDAC6HDAC3
SCHEMBL7465829 0.81 ALDH1A1 (0.37) HPGDSKDM4EALDH1A1SCN9ATLR7
SCHEMBL3065517 0.74 MAPT (0.54) ALDH1A1
SCHEMBL27609155 0.74 ALDH1A1 (0.46) HPGDSKDM4EALDH1A1TLR7L3MBTL1
SCHEMBL5201609 0.74 HPGDS (0.42) HPGDSKDM4EALDH1A1TLR7HDAC1
SCHEMBL5164159 0.73 NPC1 (0.40) KDM4EALDH1A1HDAC1L3MBTL1
SCHEMBL3062139 0.73 HTR2B (0.48) HPGDSKDM4EALDH1A1SCN9ATLR7
SCHEMBL5869050 0.71 ALDH1A1 (0.36) HPGDSKDM4EALDH1A1HPGDABCB1
SCHEMBL6608498 0.71 KDM4E (0.47) KDM4EALDH1A1
SCHEMBL5868797 0.70 CHEK1 (0.44) ALDH1A1HPGDABCB1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1224175-A2 BENZODIAZEPINE DERIVATIVES AS METABOTROPIC GLUTAMATE RECEPTOR ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2002-07-24 EP disclosed
WO-2001029012-A2 BENZODIAZEPINE DERIVATIVES AS METABOTROPIC GLUTAMATE RECEPTOR ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2001-04-26 WO disclosed