SCHEMBL5201663

SCHEMBL5201663

FC(F)(F)c1cccc(C2C=CN(CCc3ccc4cc[nH]c4c3)CC2)c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 5/20 0.39
DRD2 P14416 4/20 0.39
HTR2A P28223 2/20 0.39
TRPV6 Q9H1D0 1/20 0.37
ESR1 P03372 1/20 0.37
HTR2C P28335 2/20 0.36
BACE1 P56817 1/20 0.36
ALDH1A1 P00352 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2D6 P10635 1/20 0.35
MAPT P10636 1/20 0.35
TSHR P16473 1/20 0.35
NFKB1 P19838 1/20 0.35
MAPK1 P28482 1/20 0.35
CYP2C19 P33261 1/20 0.35
THPO P40225 1/20 0.35
MTOR P42345 1/20 0.35
BLM P54132 1/20 0.35
PMP22 Q01453 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7060315 0.86 OPRL1 (0.41) HTR1ADRD2HTR2AHTR2CALDH1A1
SCHEMBL4797430 0.81 ROCK2 (0.37) HTR1ADRD2ALDH1A1CYP1A2CYP3A4
Hydrochloric Acid SCHEMBL4589568 0.80 ROCK2 (0.37) HTR1ADRD2ALDH1A1CYP1A2CYP3A4
SCHEMBL6921067 0.76 IDE (0.41) HTR1ADRD2CYP2C19SIGMAR1
SCHEMBL11273204 0.68 HTR2C (0.46) HTR1ADRD2HTR2AHTR2C
SCHEMBL5155779 0.68 PPARG (0.50) HTR1ADRD2HTR2AHTR2CMAPT
SCHEMBL29275206 0.67 ESR1 (0.51) ESR1BACE1
SCHEMBL9422688 0.65 DRD2 (0.63) HTR1ADRD2TRPV6HTR2CALDH1A1
Hydrochloric Acid SCHEMBL9305904 0.64 DRD2 (0.62) HTR1ADRD2TRPV6HTR2CALDH1A1
SCHEMBL1401419 0.63 DRD2 (0.60) HTR1ADRD2HTR2ATRPV6HTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1383762-B1 TETRAHYDROPYRIDYL-ALKYL-HETEROCYCLES, METHOD FOR PREPARING SAME AND PHARMACEUTICAL COMPOSITIONS CONTAINING SAME SANOFI AVENTIS (FR) 2007-06-20 EP claimed