SCHEMBL6921067

SCHEMBL6921067

FC(F)(F)c1cccc(C2C=CN(CCc3cccc4ccccc34)CC2)c1

nearest known ligand 0.41

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
IDE P14735 1/20 0.41
UBE2N P61088 1/20 0.41
DRD2 P14416 2/20 0.40
MC4R P32245 1/20 0.38
SIGMAR1 Q99720 3/20 0.38
POLB P06746 1/20 0.37
CYP2C19 P33261 1/20 0.37
SLC18A2 Q05940 1/20 0.37
DRD4 P21917 2/20 0.37
GRM2 Q14416 1/20 0.37
HTR1A P08908 1/20 0.35
SLC6A4 P31645 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7060315 0.83 OPRL1 (0.41) DRD2SIGMAR1CYP2C19DRD4GRM2
SCHEMBL6921065 0.78 DRD2 (0.63) IDEUBE2NDRD2MC4RSIGMAR1
SCHEMBL4797430 0.75 ROCK2 (0.37) DRD2SIGMAR1POLBCYP2C19DRD4
SCHEMBL11273204 0.71 HTR2C (0.46) DRD2HTR1A
SCHEMBL1821251 0.65 HTR7 (0.51) DRD2DRD4HTR1A
Hydrochloric Acid SCHEMBL9486649 0.65 HTR7 (0.50) DRD2DRD4HTR1A
SCHEMBL6590789 0.64 SLC18A2 (0.46) MC4RSIGMAR1SLC18A2
SCHEMBL10475673 0.64 DRD2 (0.65) DRD2SIGMAR1DRD4GRM2
SCHEMBL30387904 0.63 HTR2C (0.37) HTR1A
SCHEMBL7951503 0.61 ADRA1D (0.48) SIGMAR1SLC18A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1357928-A4 A NOVEL PHARMACEUTICAL COMPOUND AND METHODS OF MAKING AND USING SAME NEW RIVER PHARMACEUTICALS INC (US) 2004-12-29 EP disclosed
EP-1357928-A2 A NOVEL PHARMACEUTICAL COMPOUND AND METHODS OF MAKING AND USING SAME New River Pharmaceuticals Inc. (US) 2003-11-05 EP disclosed
WO-2003020200-A2 A NOVEL PHARMACEUTICAL COMPOUND AND METHODS OF MAKING AND USING SAME NEW RIVER PHARMACEUTICALS INC. (US) 2003-03-13 WO disclosed