SCHEMBL5202185

SCHEMBL5202185

CC(C)(C)OC(=O)C(N)c1cccc(Oc2cc(Cl)ccc2NCCCC(=O)O)c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR4A2 P43354 1/20 0.39
P2RY1 P47900 1/20 0.36
SIRT5 Q9NXA8 3/20 0.36
P2RX4 Q99571 1/20 0.35
KMT2A Q03164 2/20 0.35
MEN1 O00255 1/20 0.35
MRGPRX4 Q96LA9 1/20 0.34
L3MBTL1 Q9Y468 2/20 0.34
LMNA P02545 1/20 0.34
ADRB1 P08588 1/20 0.34
ADRB3 P13945 1/20 0.34
FFAR1 O14842 2/20 0.34
PTGDR2 Q9Y5Y4 2/20 0.34
CDC25A P30304 1/20 0.34
CDC25B P30305 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
PPARG P37231 1/20 0.33
PTGER4 P35408 1/20 0.33
ALDH1A1 P00352 1/20 0.33
THRB P10828 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5202191 0.80 PPARG (0.42) FFAR1PTGDR2PPARGALDH1A1
SCHEMBL5208051 0.77 MEN1 (0.41) KMT2AMEN1LMNAPTGER4ALDH1A1
SCHEMBL5202385 0.77 MEN1 (0.41) KMT2AMEN1LMNAPTGER4ALDH1A1
SCHEMBL5206639 0.76 KDM4E (0.36) KMT2AMEN1
SCHEMBL5205373 0.74 TSPO (0.40) P2RX4FFAR1
SCHEMBL5208118 0.73 FDFT1 (0.39) P2RY1KMT2AMEN1FFAR1NPSR1
SCHEMBL5206633 0.72 KDM4E (0.40) KMT2AMEN1ALDH1A1NPSR1
SCHEMBL5205312 0.72 PPARG (0.40) PPARGALDH1A1
SCHEMBL5205112 0.71 MEN1 (0.37) P2RX4KMT2AMEN1LMNAPTGER4
SCHEMBL27637321 0.70 L3MBTL1 (0.50) L3MBTL1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7160887-B1 Aromatic amine derivatives, their production and use TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2007-01-09 US disclosed
EP-1123918-B1 AROMATIC AMINE DERIVATIVES, PROCESS FOR THE PREPARATION THEREOF AND AGENTS CONTAINING THE SAME TAKEDA PHARMACEUTICAL (JP) 2005-03-09 EP disclosed
EP-1123918-A1 AROMATIC AMINE DERIVATIVES, PROCESS FOR THE PREPARATION THEREOF AND AGENTS CONTAINING THE SAME Takeda Chemical Industries, Ltd. (JP) 2001-08-16 EP disclosed