SCHEMBL5202499

SCHEMBL5202499

CC(C)(C)OC(=O)C(N)c1cccc(Oc2ccccc2N(CCCCNC(=O)c2ccccc2F)C(=O)c2ccc(-c3ccccc3)cc2)c1

nearest known ligand 0.37

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.36
DRD2 P14416 7/20 0.36
DRD3 P35462 7/20 0.36
DRD4 P21917 1/20 0.36
ALDH1A1 P00352 1/20 0.34
MCHR1 Q99705 1/20 0.34
TDP1 Q9NUW8 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
HCRTR1 O43613 1/20 0.32
HCRTR2 O43614 1/20 0.32
PTGES O14684 1/20 0.32
ALOX5 P09917 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL5202593 0.69 TSPO (0.40) DRD2DRD3DRD4PTGESALOX5
SCHEMBL5204545 0.67 KMT2A (0.41) ALDH1A1
SCHEMBL5203387 0.67 TSPO (0.38) DRD2DRD3DRD4
SCHEMBL5203392 0.67 TSPO (0.36) DRD2DRD3DRD4
SCHEMBL5205532 0.67 TSPO (0.39) PTGESALOX5
SCHEMBL5204775 0.66 HDAC1 (0.39) PTGESALOX5
SCHEMBL5203488 0.66 TSPO (0.39) DRD2DRD3DRD4
SCHEMBL5204339 0.65 SCN9A (0.39) KDM4EALDH1A1
SCHEMBL22880704 0.64 NPC1 (0.52) ALDH1A1TDP1HCRTR1
SCHEMBL28527692 0.63 NPSR1 (0.51) KDM4EALDH1A1TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7160887-B1 Aromatic amine derivatives, their production and use TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2007-01-09 US disclosed
EP-1123918-B1 AROMATIC AMINE DERIVATIVES, PROCESS FOR THE PREPARATION THEREOF AND AGENTS CONTAINING THE SAME TAKEDA PHARMACEUTICAL (JP) 2005-03-09 EP disclosed
EP-1123918-A1 AROMATIC AMINE DERIVATIVES, PROCESS FOR THE PREPARATION THEREOF AND AGENTS CONTAINING THE SAME Takeda Chemical Industries, Ltd. (JP) 2001-08-16 EP disclosed