SCHEMBL28527692

SCHEMBL28527692

CC(C)(C)OC(=O)N[C@@H](CCCCNC(=O)c1ccccc1F)C(=O)OC(C)(C)C

nearest known ligand 0.55

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 7/20 0.51
MEN1 O00255 5/20 0.51
KMT2A Q03164 5/20 0.51
POLB P06746 4/20 0.51
TDP1 Q9NUW8 6/20 0.50
MAPT P10636 4/20 0.50
ATM Q13315 2/20 0.50
ALDH1A1 P00352 1/20 0.49
PAX8 Q06710 1/20 0.49
KDM4E B2RXH2 1/20 0.49
KLK7 P49862 1/20 0.48
KLK5 Q9Y337 1/20 0.48
CTSS P25774 1/20 0.46
CTSK P43235 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22880704 0.84 NPC1 (0.52) MEN1KMT2ATDP1ALDH1A1
SCHEMBL32665591 0.79 NPSR1 (0.53) NPSR1MEN1KMT2APOLBTDP1
SCHEMBL6379646 0.79 CTSS (0.53) CTSSCTSK
SCHEMBL31758256 0.79 TDP1 (0.61) NPSR1MEN1KMT2APOLBTDP1
SCHEMBL17309872 0.78 MAPT (0.68) NPSR1MEN1KMT2ATDP1MAPT
SCHEMBL1303931 0.78 MAPT (0.68) NPSR1MEN1KMT2ATDP1MAPT
SCHEMBL8239220 0.77 ALDH1A1 (0.57) ALDH1A1CTSK
SCHEMBL346337 0.77 ALDH1A1 (0.57) ALDH1A1CTSK
SCHEMBL32665504 0.76 KLK7 (0.54) NPSR1MEN1KMT2APOLBTDP1
SCHEMBL26862002 0.76 SIRT1 (0.56) NPSR1MEN1KMT2APOLBTDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112358414-B Unnatural amino acids and their use in protein site-directed modification and protein interactions 中国科学院上海药物研究所 2022-03-22 CN disclosed
CN-112358414-A Unnatural amino acids and their use in protein site-directed modification and protein interactions 中国科学院上海药物研究所 2021-02-12 CN disclosed