SCHEMBL5202743

SCHEMBL5202743

Cc1nccc(C(F)(F)F)c1C=O

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SORT1 Q99523 1/20 0.35
NFE2L2 Q16236 8/20 0.33
ALDH1A1 P00352 2/20 0.32
KDM4E B2RXH2 1/20 0.32
MEN1 O00255 1/20 0.32
LMNA P02545 1/20 0.32
HPGD P15428 1/20 0.32
KMT2A Q03164 1/20 0.32
AOX1 Q06278 1/20 0.32
KIF11 P52732 1/20 0.32
ERN1 O75460 2/20 0.31
SLC22A12 Q96S37 1/20 0.31
CYP1A2 P05177 2/20 0.31
CYP3A4 P08684 2/20 0.31
ALOX15 P16050 1/20 0.31
TSHR P16473 1/20 0.31
MAPK1 P28482 1/20 0.31
HIF1A Q16665 1/20 0.31
HSD17B10 Q99714 1/20 0.31
TDP1 Q9NUW8 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17255057 0.81 MEN1 (0.34) NFE2L2ALDH1A1MEN1LMNAKMT2A
SCHEMBL31028560 0.81 MEN1 (0.34) NFE2L2ALDH1A1MEN1LMNAKMT2A
SCHEMBL29954958 0.79 NOS3 (0.36) NFE2L2KIF11ERN1TSHRHSD17B10
SCHEMBL27979595 0.79 NOS3 (0.36) NFE2L2KIF11ERN1TSHRHSD17B10
SCHEMBL31711438 0.77 NFE2L2 (0.35) NFE2L2KIF11
SCHEMBL4383164 0.76 SORT1 (0.33) SORT1ALDH1A1KDM4EMEN1HPGD
SCHEMBL29953139 0.75 ERN1 (0.35) ALDH1A1KDM4EMEN1LMNAHPGD
SCHEMBL30547062 0.75 DHODH (0.35) SORT1ALDH1A1SLC22A12CYP1A2CYP3A4
SCHEMBL4383170 0.75 DHODH (0.35) SORT1ALDH1A1SLC22A12CYP1A2CYP3A4
SCHEMBL15147449 0.74 CYP1A2 (0.37) SORT1ALDH1A1SLC22A12CYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1654253-B1 SUBSTITUTED 3-PYRROLIDIN-INDOLE DERIVATIVES GRUENENTHAL GMBH (DE) 2007-01-03 EP disclosed