SCHEMBL5203345

SCHEMBL5203345

CCOC(=O)CCCNc1ccccc1Oc1ccc(CNC(=O)OC(C)(C)C)cc1

nearest known ligand 0.43

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 2/20 0.43
TOP2A P11388 1/20 0.42
LTA4H P09960 4/20 0.42
NAMPT P43490 1/20 0.41
CA1 P00915 1/20 0.41
CA2 P00918 1/20 0.41
CACNA1B Q00975 5/20 0.41
PPID Q08752 1/20 0.39
PDE5A O76074 1/20 0.39
ELANE P08246 1/20 0.39
FAAH O00519 1/20 0.38
ALOX15 P16050 1/20 0.38
KDM4E B2RXH2 1/20 0.38
MAPT P10636 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5201771 0.85 NAMPT (0.47) HDAC1TOP2ALTA4HNAMPTCA1
SCHEMBL5203338 0.81 TOP2A (0.40) TOP2ALTA4HPDE5AELANEKDM4E
SCHEMBL5205312 0.80 PPARG (0.40) TOP2AALOX15KDM4EMAPT
SCHEMBL5202903 0.77 PPARG (0.40) FAAHALOX15
SCHEMBL6376720 0.74 CYP4F2 (0.56) NAMPTCA1CA2PPIDMAPT
SCHEMBL5205300 0.74 PPARG (0.41) ALOX15KDM4E
SCHEMBL5202388 0.74 CNR1 (0.40) HDAC1KDM4EMAPT
SCHEMBL16456594 0.74 FAAH (0.56) HDAC1NAMPTFAAH
SCHEMBL7254343 0.73 ALDH1A1 (0.46) TOP2ALTA4HNAMPT
SCHEMBL8786889 0.72 MAPT (0.51) NAMPTCA1CA2PPIDMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7160887-B1 Aromatic amine derivatives, their production and use TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2007-01-09 US disclosed
EP-1123918-B1 AROMATIC AMINE DERIVATIVES, PROCESS FOR THE PREPARATION THEREOF AND AGENTS CONTAINING THE SAME TAKEDA PHARMACEUTICAL (JP) 2005-03-09 EP disclosed
EP-1123918-A1 AROMATIC AMINE DERIVATIVES, PROCESS FOR THE PREPARATION THEREOF AND AGENTS CONTAINING THE SAME Takeda Chemical Industries, Ltd. (JP) 2001-08-16 EP disclosed