SCHEMBL5203373

SCHEMBL5203373

CSc1ncccc1[C]=O

nearest known ligand 0.41

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.41
L3MBTL1 Q9Y468 4/20 0.39
RAB9A P51151 2/20 0.39
TSHR P16473 2/20 0.39
CASP3 P42574 2/20 0.39
SENP8 Q96LD8 2/20 0.39
SENP7 Q9BQF6 2/20 0.39
SENP6 Q9GZR1 2/20 0.39
KDM4E B2RXH2 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
NPC1 O15118 2/20 0.37
HPGD P15428 1/20 0.37
MEN1 O00255 1/20 0.37
TDP1 Q9NUW8 1/20 0.36
ALDH1A1 P00352 2/20 0.35
HTT P42858 1/20 0.35
GLA P06280 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1846079 0.80 TSHR (0.44) KMT2AL3MBTL1RAB9ATSHRCASP3
SCHEMBL27165240 0.80 GRM5 (0.39) KMT2AL3MBTL1RAB9ATSHRCASP3
SCHEMBL5519355 0.79 ALDH1A1 (0.41) KMT2AL3MBTL1RAB9ATSHRKDM4E
SCHEMBL7710680 0.77 HSD11B1 (0.44) L3MBTL1RAB9AKDM4ENPSR1NPC1
SCHEMBL27165246 0.76 KMT2A (0.35) KMT2AL3MBTL1RAB9ATSHRCASP3
SCHEMBL27165236 0.73 KDM4E (0.36) KMT2AL3MBTL1RAB9ATSHRCASP3
SCHEMBL1464520 0.72
SCHEMBL7524889 0.72 CYP1A2 (0.44) KMT2AL3MBTL1TSHRKDM4EHPGD
SCHEMBL10833630 0.70 L3MBTL1 (0.47) KMT2AL3MBTL1RAB9ATSHRCASP3
SCHEMBL6385617 0.70 TDP1 (0.33) KMT2AL3MBTL1TSHRKDM4ENPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1189891-A1 TRIAZOLE COMPOUNDS AND COMBINATORIAL LIBRARIES THEREOF LION Bioscience AG (DE) 2002-03-27 EP claimed
US-6362342-B1 BIOSYNTHESIS; DRUG LIBRARIES LION BIOSCIENCE AG (DE) 2002-03-26 US claimed
WO-2001000594-A1 TRIAZOLE COMPOUNDS AND COMBINATORIAL LIBRARIES THEREOF LION BIOSCIENCE AG (DE) 2001-01-04 WO claimed
EP-1654253-B1 SUBSTITUTED 3-PYRROLIDIN-INDOLE DERIVATIVES GRUENENTHAL GMBH (DE) 2007-01-03 EP disclosed
EP-1189891-A1 TRIAZOLE COMPOUNDS AND COMBINATORIAL LIBRARIES THEREOF LION Bioscience AG (DE) 2002-03-27 EP disclosed
US-6362342-B1 BIOSYNTHESIS; DRUG LIBRARIES LION BIOSCIENCE AG (DE) 2002-03-26 US disclosed
WO-2001000594-A1 TRIAZOLE COMPOUNDS AND COMBINATORIAL LIBRARIES THEREOF LION BIOSCIENCE AG (DE) 2001-01-04 WO disclosed