SCHEMBL5203967

SCHEMBL5203967

[CH]=CCC(CC)c1ccccc1

nearest known ligand 0.43

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
LMNA P02545 3/20 0.43
CCR5 P51681 1/20 0.41
TAAR1 Q96RJ0 4/20 0.37
CYP2D6 P10635 1/20 0.37
MIF P14174 1/20 0.36
HSD17B10 Q99714 1/20 0.36
TRPA1 O75762 3/20 0.35
HKDC1 Q2TB90 1/20 0.35
HTR2A P28223 1/20 0.34
HRH1 P35367 1/20 0.34
AOC3 Q16853 1/20 0.34
NOS3 P29474 1/20 0.34
NOS2 P35228 1/20 0.34
CTSD P07339 1/20 0.34
CTSE P14091 1/20 0.34
BACE1 P56817 1/20 0.34
POLB P06746 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5207585 0.84 AOC3 (0.40) LMNACCR5TRPA1HTR2AHRH1
SCHEMBL5202807 0.81 POLB (0.40) LMNAHTR2AHRH1AOC3POLB
SCHEMBL1111815 0.81 LMNA (0.45) LMNACCR5TAAR1CYP2D6MIF
SCHEMBL7384257 0.80 LMNA (0.41) LMNACCR5TAAR1CYP2D6MIF
SCHEMBL8121030 0.80 NR1I2 (0.39) HTR2APOLB
SCHEMBL169508 0.79 LMNA (0.56) LMNACCR5TAAR1CYP2D6MIF
SCHEMBL4901936 0.79 CYP2C19 (0.48) LMNACCR5TAAR1CYP2D6MIF
SCHEMBL4864892 0.79 CCR5 (0.45) LMNACCR5TAAR1CYP2D6MIF
SCHEMBL464510 0.79 CCR5 (0.45) LMNACCR5TAAR1CYP2D6MIF
SCHEMBL2133730 0.79 CYP2C19 (0.48) LMNACCR5TAAR1CYP2D6MIF

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0980867-B1 KETONE DERIVATIVES AND MEDICINAL USE THEREOF TORAY INDUSTRIES (JP) 2007-08-08 EP disclosed
CN-1114602-C Ketone derivatives and medicinal use thereof TORAY INDUSTRIES (JP) 2003-07-16 CN disclosed
US-6100292-A Ketone derivatives and their medical applications TORAY INDUSTRIES, INC. (JP) 2000-08-08 US disclosed
EP-0980867-A1 KETONE DERIVATIVES AND MEDICINAL USE THEREOF TORAY INDUSTRIES, INC. (JP) 2000-02-23 EP disclosed
CN-1242771-A Ketone derivatives and medicinal use thereof TORAY INDUSTRIES (JP) 2000-01-26 CN disclosed
CN-1039321-C New beta-amino-alpha-hydroxycarboxylic acids and their use SANKYO CO (JP) 1998-07-29 CN disclosed
CN-1064683-A New beta-amino-alpha-hydroxycarboxylic acids and uses thereof SANKYO CO (JP) 1992-09-23 CN disclosed
EP-0498680-A1 New beta-amino-alpha-hydroxycarboxylic acids and their use Sankyo Company Limited (JP) 1992-08-12 EP disclosed