SCHEMBL5204620

SCHEMBL5204620

Cc1cnc(-c2ccc(C(F)(F)F)cc2)nc1C

nearest known ligand 0.45

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.45
THRB P10828 1/20 0.45
TRPV3 Q8NET8 5/20 0.42
KIF11 P52732 3/20 0.41
SORT1 Q99523 1/20 0.41
S1PR1 P21453 3/20 0.40
KCNH2 Q12809 1/20 0.40
TDP2 O95551 1/20 0.39
ADORA3 P0DMS8 1/20 0.38
GABBR2 O75899 1/20 0.38
GABBR1 Q9UBS5 1/20 0.38
HEXA P06865 1/20 0.38
HEXB P07686 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12538714 0.85 TRPV3 (0.50) LMNATHRBTRPV3KIF11S1PR1
SCHEMBL25979339 0.84 NPC1 (0.49) LMNAKIF11
SCHEMBL5219754 0.83 LMNA (0.43) LMNATHRBTRPV3KIF11S1PR1
SCHEMBL5249070 0.83 TRPV3 (0.43) LMNATHRBTRPV3KIF11ADORA3
SCHEMBL27942884 0.83 DPP4 (0.46) LMNATHRBTRPV3KIF11S1PR1
SCHEMBL14983666 0.81 IDO1 (0.47)
SCHEMBL14983674 0.80 NPC1 (0.42) LMNAKCNH2
SCHEMBL6017152 0.80 TRPV3 (0.46) LMNATHRBTRPV3KCNH2
SCHEMBL1549695 0.80 KCNH2 (0.41) LMNATHRBTRPV3KIF11S1PR1
SCHEMBL5202727 0.80 TRPV3 (0.46) LMNATHRBTRPV3KIF11S1PR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1036066-B1 SUBSTITUTED PYRIMIDINE AND PYRIDINE HERBICIDES MID AMERICA COMMERCIALIZATION (US) 2007-04-18 EP disclosed
US-20040033896-A1 E.g., 5-ethyl-4-((3 -(trifluoromethoxy)phenyl)methyl)-2-(3-(trifluoromethyl)-1H pyrazol-1-yl)pyrimidine and 5-methyl-2-(4-(trifluoromethyl)phenyl)-4-((3-(trifluoromethyl) phenyl)methyl)pyrimidine KOETHER GERARD (US) 2004-02-19 US disclosed
US-6525001-B1 5-methyl-2-(4-(trifluoromethyl)phenyl)-4-((3 -(trifluoromethyl)phenyl)methyl)pyrimidine MID-AMERICAN COMMERCIALIZATION CORPORATION 2003-02-25 US disclosed
EP-1036066-A1 SUBSTITUTED PYRIMIDINE AND PYRIDINE HERBICIDES E.I. DU PONT DE NEMOURS AND COMPANY (US) 2000-09-20 EP disclosed
WO-1999028301-A1 SUBSTITUTED PYRIMIDINE AND PYRIDINE HERBICIDES E.I. DU PONT DE NEMOURS AND COMPANY (US) 1999-06-10 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040033896-A1 E.g., 5-ethyl-4-((3 -(trifluoromethoxy)phenyl)methyl)-2-(3-(trifluoromethyl)-1H pyrazol-1-yl)pyrimidine and 5-methyl-2-(4-(trifluoromethyl)phenyl)-4-((3-(trifluoromethyl) phenyl)methyl)pyrimidine PYM1, Q6ZSR9, MRM1 LMNA 3056/4885THRB 3346/4885TRPV3 3202/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.