SCHEMBL5204638

SCHEMBL5204638

CN(Cc1ccccc1)CC1CCCCC1(O)c1cccnc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 9/20 0.47
SLC6A2 P23975 9/20 0.47
SLC6A4 P31645 9/20 0.47
OPRD1 P41143 3/20 0.47
OPRK1 P41145 3/20 0.47
MEN1 O00255 3/20 0.47
KMT2A Q03164 3/20 0.47
SLC22A1 O15245 2/20 0.45
CHRM2 P08172 2/20 0.45
CHRM1 P11229 2/20 0.45
OPRL1 P41146 2/20 0.44
CNR2 P34972 1/20 0.41
SLC6A9 P48067 1/20 0.41
CHRNB2 P17787 1/20 0.39
CHRNA4 P43681 1/20 0.39
ALDH1A1 P00352 2/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
CHRM4 P08173 1/20 0.39
CHRM5 P08912 1/20 0.39
CHRM3 P20309 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL4864830 1.00 OPRM1 (0.47) OPRM1SLC6A2SLC6A4OPRD1OPRK1
Hydrochloric Acid SCHEMBL4859953 0.86 SLC6A4 (0.62) OPRM1SLC6A2SLC6A4OPRD1OPRK1
SCHEMBL5205111 0.85 SLC6A4 (0.64) OPRM1SLC6A2SLC6A4OPRD1OPRK1
SCHEMBL6167477 0.84 SLC6A4 (0.62) OPRM1SLC6A2SLC6A4OPRD1OPRK1
SCHEMBL5880618 0.81 SLC6A4 (0.58) OPRM1SLC6A2SLC6A4OPRD1OPRK1
SCHEMBL5880531 0.81 SLC6A2 (0.43) OPRM1SLC6A2SLC6A4OPRD1OPRK1
SCHEMBL11150421 0.79 SLC6A2 (0.74) OPRM1SLC6A2SLC6A4OPRD1OPRK1
SCHEMBL5880615 0.79 SLC6A2 (0.47) OPRM1SLC6A2SLC6A4OPRD1OPRK1
SCHEMBL29950758 0.78 TRPA1 (0.45) OPRM1SLC6A2SLC6A4OPRD1OPRK1
SCHEMBL28849444 0.78 TRPA1 (0.45) OPRM1SLC6A2SLC6A4OPRD1OPRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2006523182-A 2006-10-12 JP claimed
EP-1572653-A1 SATURATED AND UNSATURATED HETEROARYLCYCLOALKYLMETHYL AMINES AS ANTI-DEPRESSANTS Grünenthal GmbH (DE) 2005-09-14 EP claimed
WO-2004063161-A1 SATURATED AND UNSATURATED HETEROARYLCYCLOALKYLMETHYL AMINES AS ANTI-DEPRESSANTS Grünenthal GmbH (DE) 2004-07-29 WO claimed
EP-1572653-B1 SATURATED AND UNSATURATED HETEROARYLCYCLOALKYLMETHYL AMINES AS ANTI-DEPRESSANTS GRUENENTHAL GMBH (DE) 2007-11-21 EP disclosed
EP-1572653-A1 SATURATED AND UNSATURATED HETEROARYLCYCLOALKYLMETHYL AMINES AS ANTI-DEPRESSANTS Grünenthal GmbH (DE) 2005-09-14 EP disclosed
WO-2004063161-A1 SATURATED AND UNSATURATED HETEROARYLCYCLOALKYLMETHYL AMINES AS ANTI-DEPRESSANTS Grünenthal GmbH (DE) 2004-07-29 WO disclosed