SCHEMBL5204923

SCHEMBL5204923

O=C(O)C1=Cc2cc(-c3ccc(N4CCCC4)cc3)ccc2CCC1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 9/20 0.52
CXCR3 P49682 3/20 0.39
CXCR5 P32302 1/20 0.39
IP6K1 Q92551 2/20 0.39
DHODH Q02127 1/20 0.39
ALDH1A1 P00352 3/20 0.38
HPGD P15428 3/20 0.38
NPC1 O15118 3/20 0.38
RAB9A P51151 3/20 0.38
TP53 P04637 2/20 0.38
MAPT P10636 2/20 0.38
TSHR P16473 2/20 0.38
HSD17B10 Q99714 2/20 0.38
LMNA P02545 1/20 0.38
ALOX15 P16050 1/20 0.38
STAT1 P42224 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
CHEK1 O14757 1/20 0.38
CCR2 P41597 3/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5210006 0.99 CCR5 (0.52) CCR5CXCR3CXCR5IP6K1DHODH
SCHEMBL3499816 0.81 CCR5 (0.53) CCR5CXCR3CXCR5ALDH1A1NPC1
SCHEMBL5212207 0.79 CCR5 (0.41) CCR5IP6K1ALDH1A1HPGDNPC1
SCHEMBL7929509 0.78 KDM4E (0.37) CCR5IP6K1DHODHALDH1A1HPGD
SCHEMBL5206221 0.78 LMNA (0.43) CCR5IP6K1DHODHALDH1A1HPGD
Hydrochloric Acid SCHEMBL7968862 0.77 KDM4E (0.36) CCR5IP6K1DHODHALDH1A1HPGD
SCHEMBL7934206 0.77 DHODH (0.38) CCR5IP6K1DHODHALDH1A1HPGD
SCHEMBL5208461 0.75 CCR5 (0.53) CCR5CXCR3CXCR5NPC1RAB9A
SCHEMBL3498958 0.75 CCR5 (0.53) CCR5
SCHEMBL5209485 0.74 BCL2L1 (0.44) CCR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1040103-B1 ANILIDE DERIVATIVE, PRODUCTION AND USE THEREOF TAKEDA PHARMACEUTICAL (JP) 2007-03-14 EP disclosed
US-6413947-B1 Anilide derivative, production and use thereof TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2002-07-02 US disclosed
US-6376536-B1 VIRICIDES TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2002-04-23 US disclosed
US-6268354-B1 Pharmaceutical composition for antagonizing CCR5 comprising anilide derivative TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-07-31 US disclosed
US-6172061-B1 AIDS THERAPY TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-01-09 US disclosed
US-6166006-A Anilide derivative, production and use thereof TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2000-12-26 US disclosed
US-6096780-A ANTIVIRAL COMPOUND USEFUL FOR TREATING HIV VIRUSES TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2000-08-01 US disclosed