SCHEMBL7929509

SCHEMBL7929509

O=C(O)C1=Cc2cc(-c3ccc(N4CCCC4)cc3)ccc2S(=O)(=O)CC1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.37
DHODH Q02127 1/20 0.36
IP6K1 Q92551 2/20 0.36
CHEK1 O14757 1/20 0.36
CCR5 P51681 4/20 0.35
ALDH1A1 P00352 4/20 0.35
HPGD P15428 4/20 0.35
NPC1 O15118 4/20 0.35
RAB9A P51151 4/20 0.35
MAPT P10636 3/20 0.35
HSD17B10 Q99714 3/20 0.35
TP53 P04637 2/20 0.35
TSHR P16473 2/20 0.35
L3MBTL1 Q9Y468 2/20 0.35
ALOX15 P16050 2/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
LMNA P02545 1/20 0.35
STAT1 P42224 1/20 0.35
IP6K3 Q96PC2 1/20 0.35
IP6K2 Q9UHH9 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7934206 0.99 DHODH (0.38) KDM4EDHODHIP6K1CHEK1CCR5
Hydrochloric Acid SCHEMBL7968862 0.99 KDM4E (0.36) KDM4EDHODHIP6K1CHEK1CCR5
SCHEMBL7929505 0.91 KMO (0.39) KDM4EALDH1A1MAPTHSD17B10
Hydrochloric Acid SCHEMBL7971793 0.90 AOC3 (0.40) KDM4EALDH1A1MAPTHSD17B10L3MBTL1
SCHEMBL7959102 0.87 ALDH1A1 (0.42) KDM4ECCR5ALDH1A1HPGDNPC1
SCHEMBL7972710 0.86 ALDH1A1 (0.41) KDM4ECCR5ALDH1A1NPC1RAB9A
SCHEMBL7974920 0.83 BCL2L1 (0.39) KDM4EHSD17B10SMN1; SMN2LMNAKMT2A
SCHEMBL7929501 0.82 MCL1 (0.39) DHODHCCR5NPC1RAB9AMAPT
SCHEMBL3499284 0.82 ALAD (0.35) POLBCYP1A2CYP3A4CYP2C9
SCHEMBL7970423 0.80 HAO1 (0.35) DHODHCCR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1140896-A1 BENZOTHIEPIN-ANILIDE DERIVATIVES, THEIR PRODUCTION AND THEIR USE FOR ANTAGONIZING CCR-5 Takeda Chemical Industries, Ltd. (JP) 2001-10-10 EP disclosed
US-6235771-B1 AIDS THERPAY TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-05-22 US disclosed
WO-2000037455-A1 BENZOTHIEPIN-ANILIDE DERIVATIVES, THEIR PRODUCTION AND THEIR USE FOR ANTAGONIZING CCR-5 TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2000-06-29 WO disclosed