SCHEMBL5205002

SCHEMBL5205002

O=C(O)NCc1ccc(Oc2ccccc2NCc2ccc(-c3ccccc3)cc2)cc1

nearest known ligand 0.52

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CACNA1B Q00975 8/20 0.52
ADAMTS5 Q9UNA0 3/20 0.48
NPC1 O15118 1/20 0.48
RAB9A P51151 1/20 0.48
ALDH1A1 P00352 3/20 0.46
GAA P10253 2/20 0.46
L3MBTL1 Q9Y468 2/20 0.46
HPGD P15428 1/20 0.46
HTT P42858 1/20 0.46
ATM Q13315 1/20 0.46
LMNA P02545 1/20 0.46
MAPK14 Q16539 1/20 0.45
MEN1 O00255 1/20 0.45
KMT2A Q03164 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6174370 0.83 CACNA1B (0.48) CACNA1BADAMTS5ALDH1A1GAAL3MBTL1
SCHEMBL5205589 0.80 CACNA1B (0.50) CACNA1BNPC1RAB9AALDH1A1LMNA
SCHEMBL7834277 0.79 FFAR1 (0.44) ADAMTS5RAB9AALDH1A1GAAL3MBTL1
SCHEMBL1730117 0.78 LMNA (0.68) NPC1RAB9AALDH1A1GAAHTT
SCHEMBL5206113 0.78 ADAMTS5 (0.48) ADAMTS5NPC1RAB9AALDH1A1GAA
SCHEMBL7242067 0.77 FFAR1 (0.54) ADAMTS5ALDH1A1HPGDLMNAMEN1
SCHEMBL1728537 0.77 MAPK14 (0.68) ALDH1A1GAAL3MBTL1HPGDHTT
SCHEMBL11215406 0.77 CACNA1B (0.63) CACNA1BGAAL3MBTL1HPGD
SCHEMBL6178139 0.77 CYP1A2 (0.51) NPC1ALDH1A1GAAL3MBTL1HPGD
SCHEMBL11216479 0.75 CACNA1B (0.58) CACNA1BGAAHTTATMMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7160887-B1 Aromatic amine derivatives, their production and use TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2007-01-09 US disclosed