SCHEMBL5205589

SCHEMBL5205589

CC(C)(C)N(Cc1ccc(Oc2ccccc2NCc2ccc(-c3ccccc3)cc2)cc1)C(=O)O

nearest known ligand 0.50

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CACNA1B Q00975 12/20 0.50
ALDH1A1 P00352 1/20 0.42
KDM4C Q9H3R0 2/20 0.42
KDM5B Q9UGL1 1/20 0.41
LMNA P02545 1/20 0.40
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5205144 0.91 CACNA1B (0.44) CACNA1BLMNAMEN1KMT2A
SCHEMBL5203690 0.82 FFAR1 (0.47) ALDH1A1KDM4CKDM5BLMNAMEN1
SCHEMBL5204934 0.81 PTGES (0.39) KDM4CKDM5BMEN1KMT2A
SCHEMBL5205774 0.81 ADAMTS5 (0.40) ALDH1A1MEN1KMT2A
SCHEMBL5205002 0.80 CACNA1B (0.52) CACNA1BALDH1A1LMNANPC1RAB9A
SCHEMBL5201809 0.78 FFAR1 (0.49) CACNA1B
SCHEMBL5206544 0.77 MEN1 (0.45) ALDH1A1LMNAMEN1KMT2A
SCHEMBL6174370 0.76 CACNA1B (0.48) CACNA1BALDH1A1KDM4CKDM5BLMNA
SCHEMBL5202945 0.73 ALDH1A1 (0.48) ALDH1A1LMNANPC1RAB9AMEN1
SCHEMBL4019172 0.73 MAPK14 (0.67) LMNANPC1RAB9AMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7160887-B1 Aromatic amine derivatives, their production and use TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2007-01-09 US disclosed