SCHEMBL5206068

SCHEMBL5206068

CC(Oc1ccccc1)C(=O)N1CCC(c2cn(Cc3ccc(C#N)cc3)c3ccccc23)C1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.49
HTT P42858 2/20 0.49
SMO Q99835 1/20 0.49
CNR2 P34972 1/20 0.46
POLB P06746 1/20 0.44
HRH2 P25021 2/20 0.43
HDAC3 O15379 1/20 0.43
HDAC1 Q13547 1/20 0.43
HDAC2 Q92769 1/20 0.43
HDAC10 Q969S8 1/20 0.43
HDAC8 Q9BY41 1/20 0.43
HDAC6 Q9UBN7 1/20 0.43
NCOR2 Q9Y618 1/20 0.43
NPSR1 Q6W5P4 2/20 0.41
MAPT P10636 1/20 0.41
DRD2 P14416 1/20 0.41
HTR6 P50406 1/20 0.41
THRB P10828 2/20 0.41
HTR2A P28223 2/20 0.40
HTR2C P28335 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5202142 0.85 LMNA (0.50) LMNAHTTSMOCNR2POLB
SCHEMBL4859761 0.84 HRH2 (0.48) HRH2MAPTHTR2AHTR2CHTR2B
SCHEMBL5203814 0.82 SMO (0.51) LMNAHTTSMOCNR2POLB
SCHEMBL4852063 0.81 HRH2 (0.53) HRH2THRBHTR2AHTR2CHTR2B
SCHEMBL5205062 0.75 SMO (0.46) LMNAHTTSMOCNR2POLB
SCHEMBL3598410 0.74 SMO (0.54) LMNAHTTSMOCNR2POLB
SCHEMBL5203146 0.74 SMO (0.47) LMNAHTTSMOCNR2POLB
SCHEMBL5203143 0.72 CNR2 (0.43) LMNAHTTSMOCNR2POLB
SCHEMBL13445248 0.71 SMO (0.57) SMOCNR2HRH2NPSR1DRD2
SCHEMBL4859500 0.71 KMT2A (0.52) LMNAHTTSMOPOLBHRH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1654253-B1 SUBSTITUTED 3-PYRROLIDIN-INDOLE DERIVATIVES GRUENENTHAL GMBH (DE) 2007-01-03 EP claimed
EP-1654253-B1 SUBSTITUTED 3-PYRROLIDIN-INDOLE DERIVATIVES GRUENENTHAL GMBH (DE) 2007-01-03 EP disclosed